Identification of signalling components in tyrosine kinase cascades using phosphopeptide affinity chromatography

Biochem Biophys Res Commun. 1997 May 29;234(3):748-53. doi: 10.1006/bbrc.1997.6702.

Abstract

Various methods are now available to identify the molecular partners of the component of a signal transduction pathway. Some interactions, however, can be technically difficult to detect because they depend upon transient tyrosine phosphorylation. Here, we present a simple affinity chromatography approach based on synthetic phosphopeptides to purify potential partners of phosphotyrosine-containing proteins. With this approach, we confirm the previously characterized interaction between Grb2 and the EGF receptor, and we identify novel partners of the IGF-1 receptor and of the JAK proteins. Methenyltetrahydrofolate synthetase (MTHFS) was identified as a potential mediator of IGF-1R dependent transformation. P85alpha, the regulatory subunit of PI3 kinase, was identified as one of four proteins recruited by a phosphopeptide mimicking a motif conserved in all JAK family members.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adaptor Proteins, Signal Transducing*
  • Amino Acid Sequence
  • Animals
  • Chromatography, Affinity / methods*
  • ErbB Receptors / metabolism
  • GRB2 Adaptor Protein
  • HL-60 Cells
  • Humans
  • Molecular Sequence Data
  • Phosphopeptides / chemistry*
  • Phosphorylation
  • Protein Binding
  • Protein-Tyrosine Kinases / chemistry
  • Protein-Tyrosine Kinases / metabolism*
  • Proteins / metabolism
  • Receptor, IGF Type 1 / metabolism
  • Sequence Homology, Amino Acid
  • Signal Transduction*

Substances

  • Adaptor Proteins, Signal Transducing
  • GRB2 Adaptor Protein
  • GRB2 protein, human
  • Phosphopeptides
  • Proteins
  • ErbB Receptors
  • Protein-Tyrosine Kinases
  • Receptor, IGF Type 1