Cooperation between the Fc epsilonR1 and formyl peptide receptor signaling pathways in RBL(FPR) cells: the contribution of receptor-specific Ca2+ mobilization responses

Biochem Biophys Res Commun. 1997 Jun 27;235(3):812-9. doi: 10.1006/bbrc.1997.6874.

Abstract

RBL(FPR) mast cells express the tyrosine kinase-coupled IgE receptor, Fc epsilonR1, and the G-protein-coupled formyl peptide receptor, FPR. Fc epsilonR1 crosslinking causes Ca2+ stores release, Ca2+ influx, Ins(1,4,5)P3 production and secretion. FPR ligation also mobilizes Ca2+, but without measurable Ins(1,4,5)P3 production or secretion. Co-stimulating the FPR and Fc epsilonR1 induces more Ins(1,4,5)P3 production and secretion than Fc epsilonR1 cross-linking alone. Costimulation also produces more rapid and sustained Ca2+ responses than are generated by Fc epsilonR1 activation alone. We identified multiple differences between the FPR- and Fc epsilonR1-coupled Ca2+ responses, including a more rapid Ca2+ spike response to FPR ligation; intracellular Ca2+ stores that are empty following Fc epsilonR1 crosslinking but partially full following FPR activation; a more sustained Ca2+ influx response to Fc epsilonR1 crosslinking; and the immediate inhibition of stimulated Ca2+ influx by FPR antagonists but not by monovalent ligand that terminates Fc epsilonR1 crosslinking. We hypothesize that the interaction of receptor-specific Ca2+ mobilization pathways contributes to the FPR-mediated potentiation of Fc epsilonR1-coupled secretion.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Calcium / metabolism*
  • Cross-Linking Reagents
  • Dinitrophenols / pharmacology
  • HL-60 Cells
  • Humans
  • Immunoglobulin E / pharmacology
  • Inositol 1,4,5-Trisphosphate / metabolism*
  • Kinetics
  • N-Formylmethionine Leucyl-Phenylalanine / pharmacology*
  • Rats
  • Receptor Protein-Tyrosine Kinases / metabolism
  • Receptors, Formyl Peptide
  • Receptors, IgE / biosynthesis
  • Receptors, IgE / physiology*
  • Receptors, Immunologic / biosynthesis
  • Receptors, Immunologic / physiology*
  • Receptors, Peptide / biosynthesis
  • Receptors, Peptide / physiology*
  • Recombinant Fusion Proteins / metabolism
  • Serum Albumin, Bovine / pharmacology
  • Signal Transduction*
  • Thapsigargin / pharmacology
  • Transfection
  • Tumor Cells, Cultured

Substances

  • Cross-Linking Reagents
  • Dinitrophenols
  • Receptors, Formyl Peptide
  • Receptors, IgE
  • Receptors, Immunologic
  • Receptors, Peptide
  • Recombinant Fusion Proteins
  • dinitrophenyl-bovine serum albumin
  • Serum Albumin, Bovine
  • Immunoglobulin E
  • N-Formylmethionine Leucyl-Phenylalanine
  • Thapsigargin
  • Inositol 1,4,5-Trisphosphate
  • Receptor Protein-Tyrosine Kinases
  • Calcium