Indomethacin depresses prostaglandin F2 alpha-induced contraction in guinea-pig uterine artery with both intact and denuded endoth

Prostaglandins. 1997 Jun;53(6):371-9. doi: 10.1016/s0090-6980(97)00055-5.

Abstract

The purpose of this study was to explore whether cyclooxygenase products derived from endothelium or vascular muscle participate in the response of guinea-pig uterine arterial rings to prostaglandin F2 alpha (PGF2 alpha). Contraction to PGF2 alpha (0.1-30 microM) occurred with and without endothelium at similar potency and efficacy (pEC50 (-log EC50) values respectively 5.87 +/- 0.06 and 5.97 +/- 0.07; maximal response respectively 78.1 +/- 1.3% and 76.9 +/- 1.5% of contraction induced by 126 mM KCl). Indomethacin (3-30 microM) suppressed the maximum response to PGF2 alpha and induced a rightward shift of concentration-response curves, regardless of the presence of endothelium. pIC50 values for indomethacin were 4.67 and 4.74 for vessels with and without endothelium, respectively. In contrast, the thromboxane synthesis inhibitor OKY-046 (10 and 100 microM) did not affect the response to PGF2 alpha. We conclude that the PGF2 alpha-induced contraction in guinea-pig uterine artery is mediated, at least in part, through constrictor non-thromboxane prostanoid(s) of vascular muscle origin.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Arteries / physiology
  • Cyclooxygenase Inhibitors / pharmacology*
  • Dinoprost / pharmacology*
  • Endothelium, Vascular / physiology*
  • Enzyme Inhibitors / pharmacology
  • Female
  • Guinea Pigs
  • Indomethacin / pharmacology*
  • Methacrylates / pharmacology
  • Muscle, Smooth, Vascular / physiology
  • Thromboxane-A Synthase / antagonists & inhibitors
  • Uterine Contraction / drug effects*
  • Uterus / blood supply*

Substances

  • Cyclooxygenase Inhibitors
  • Enzyme Inhibitors
  • Methacrylates
  • Dinoprost
  • Thromboxane-A Synthase
  • ozagrel
  • Indomethacin