Abstract
Using immunoprecipitation and phosphotyrosine detection by Western blotting, intracellular signaling intermediates were analyzed in human primary dermal fibroblasts, either seeded as monolayers on collagen I coats (2D) or seeded within three-dimensional collagen I lattices (3D). Previous results demonstrated that integrin activation in these systems resulted in a cascade of protein tyrosine phosphorylation, including focal adhesion kinase (D. Roeckel and T. Krieg, 1994, Exp. Cell Res. 211, 42-48). Further downstream signaling events are now shown to include coordinate activation of ERK1 and ERK2 at 2 h after cell-collagen contact, irrespective of 2D or 3D culture conditions. Applying U-73122, an inhibitor of PLC, inhibits collagen lattice contraction in a dose-dependent fashion. Immunoprecipitation identified the isoform PLCgamma-1 as playing a role as signaling intermediate in fibroblast-collagen interactions. PLCgamma-1 becomes phosphorylated within 10 min after culture initiation and declines after 2 h. So far, no qualitative differences in signaling intermediates between 2D and 3D cultures have been identified.
Publication types
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Research Support, Non-U.S. Gov't
MeSH terms
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Calcium-Calmodulin-Dependent Protein Kinases / metabolism*
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Cell Adhesion
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Cell Culture Techniques / methods
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Collagen
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Enzyme Activation
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Enzyme Inhibitors / pharmacology
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Estrenes / pharmacology
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Extracellular Matrix / physiology*
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Fibroblasts / cytology
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Fibroblasts / drug effects
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Fibroblasts / physiology
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Humans
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Isoenzymes / antagonists & inhibitors
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Isoenzymes / metabolism*
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Mitogen-Activated Protein Kinase 1
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Mitogen-Activated Protein Kinase 3
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Mitogen-Activated Protein Kinases*
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Phospholipase C gamma
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Phosphorylation
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Phosphotyrosine / metabolism*
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Pyrrolidinones / pharmacology
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Skin / cytology*
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Skin Physiological Phenomena*
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Type C Phospholipases / antagonists & inhibitors
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Type C Phospholipases / metabolism*
Substances
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Enzyme Inhibitors
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Estrenes
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Isoenzymes
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Pyrrolidinones
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1-(6-((3-methoxyestra-1,3,5(10)-trien-17-yl)amino)hexyl)-1H-pyrrole-2,5-dione
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Phosphotyrosine
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Collagen
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Calcium-Calmodulin-Dependent Protein Kinases
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Mitogen-Activated Protein Kinase 1
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Mitogen-Activated Protein Kinase 3
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Mitogen-Activated Protein Kinases
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Type C Phospholipases
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Phospholipase C gamma