Vascular effects of PTHrP (1-34) and PTH (1-34) in the human fetal-placental circulation

Placenta. 1997 Sep;18(7):587-92. doi: 10.1016/0143-4004(77)90014-5.

Abstract

The aim of this study was to examine the vasodilatory effects of parathyroid hormone-related protein (PTHrP) (1-34) and parathyroid hormone (PTH) (1-34) on the human fetal-placental circulation utilising an in vitro placental perfusion model. In all experiments, the vasculature of an isolated human placental cotyledon was pre-constricted with the thromboxane A2 mimetic U46619. A simple dose of PTHrP (1-34) or PTH (1-34) (1.7-300 nM) was then infused into the fetal-placental circulation of the cotyledon. In other experiments, cotyledons were repeatedly infused with PTHrP (1-34) or PTH (1-34) (51.3 nM). Vasodilatory responses were significantly reduced in response to repeated exposure to PTHrP (1-34) (P < 0.001), indicating that this peptide desensitizes the fetal-placental vasculature. PTHrP (1-34) and PTH (1-34) equipotently stimulated a significant vasodilation of the fetal-placental circulation (P < 0.0001). The PTHrP receptor antagonist [Asn10, Leu 11]PTHrP (7-34) (102 nM) was infused in U46619-constricted placentae in the presence and absence of PTHrP (1-34) (10.2 nM). The PTHrP antagonist alone had no significant effect in the fetal-placental circulation. The antagonist significantly attenuated the response to PTHrP (1-34) (P < 0.015). Based on the data obtained in this study it is suggested that locally produced PTHrP (1-34) may be involved in the regulation of normal human fetal-placental vascular tone in autocrine and/or paracrine fashion.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid
  • Female
  • Fetus / blood supply*
  • Humans
  • Parathyroid Hormone-Related Protein*
  • Peptide Fragments / administration & dosage
  • Peptide Fragments / pharmacology*
  • Placenta / blood supply*
  • Placenta / drug effects
  • Pregnancy
  • Prostaglandin Endoperoxides, Synthetic / pharmacology
  • Proteins / administration & dosage
  • Proteins / pharmacology*
  • Receptor, Parathyroid Hormone, Type 1
  • Receptors, Parathyroid Hormone / antagonists & inhibitors
  • Teriparatide / administration & dosage
  • Teriparatide / pharmacology*
  • Thromboxane A2 / analogs & derivatives
  • Thromboxane A2 / pharmacology
  • Vasoconstrictor Agents / pharmacology
  • Vasodilation / drug effects

Substances

  • Parathyroid Hormone-Related Protein
  • Peptide Fragments
  • Prostaglandin Endoperoxides, Synthetic
  • Proteins
  • Receptor, Parathyroid Hormone, Type 1
  • Receptors, Parathyroid Hormone
  • Vasoconstrictor Agents
  • Teriparatide
  • parathyroid hormone-related protein (1-34)
  • Thromboxane A2
  • 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid