Evidence that certain 8-aminoquinolines are potentially effective drugs against Chagas disease

Ann Trop Med Parasitol. 1997 Mar;91(2):147-52. doi: 10.1080/00034983.1997.11813124.

Abstract

Forty 8-aminoquinolines (a chemical class with members having some activity against Trypanosoma cruzi infections) were evaluated for their effectiveness in reducing the 14-day parasitaemias of 4-6 week-old, female, albino mice infected with a Brazilian strain of T. cruzi. Six of the compounds were more active or as active as the reference drug, nifurtimox, and one was > 13-fold as efficacious. Certain members of the series tested warrant further evaluation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aminoquinolines / therapeutic use*
  • Animals
  • Antiparasitic Agents / therapeutic use
  • Chagas Disease / drug therapy*
  • Drug Evaluation, Preclinical
  • Female
  • Mice
  • Nifurtimox / therapeutic use
  • Parasitemia / drug therapy*

Substances

  • Aminoquinolines
  • Antiparasitic Agents
  • Nifurtimox