Trifluoroethanol induces the self-association of specific amphipathic peptides

FEBS Lett. 1997 Oct 27;416(3):265-8. doi: 10.1016/s0014-5793(97)01224-6.

Abstract

We have examined the effect of trifluoroethanol (TFE) on the solution behaviour of three amphipathic peptides. One of the peptides, containing three heptad repeat units (Ac-YS-(AKEAAKE)3GAR-NH2), remained monomeric under conditions where TFE induced a two-state transition from a random coil to an alpha-helix. In contrast, the TFE-induced alpha-helical formation of two peptides derived from human apolipoproteins C-II and E was accompanied by the formation of discrete dimers and trimers, respectively. The apolipoprotein C-II peptide further aggregated to form beta-sheet at higher concentrations of TFE (50% v/v). The results suggest a class of peptides capable of discrete self-association in the presence of cosolvents which favour intramolecular hydrogen bonding.

MeSH terms

  • Amino Acid Sequence
  • Apolipoprotein C-II
  • Apolipoproteins C / chemistry*
  • Apolipoproteins C / drug effects
  • Apolipoproteins E / chemistry*
  • Apolipoproteins E / drug effects
  • Circular Dichroism
  • Humans
  • Hydrogen Bonding
  • Molecular Sequence Data
  • Peptide Fragments / chemistry*
  • Peptide Fragments / drug effects
  • Peptides / chemistry*
  • Peptides / drug effects
  • Protein Structure, Secondary*
  • Trifluoroethanol / pharmacology*
  • Viscosity

Substances

  • Apolipoprotein C-II
  • Apolipoproteins C
  • Apolipoproteins E
  • Peptide Fragments
  • Peptides
  • Trifluoroethanol