Pharmacological studies on Puerariae flos III: protective effects of kakkalide on ethanol-induced lethality and acute hepatic injury in mice

J Pharm Pharmacol. 1997 Aug;49(8):831-3. doi: 10.1111/j.2042-7158.1997.tb06122.x.

Abstract

Kakkalide, one of the major isoflavonoid components of Puerariae flos, has been investigated for its effect on ethanol-induced intoxication and on hepatic injury, including hyperglycaemia, in mice. Kakkalide reduced mortality associated with administration of ethanol. At doses of 100 and 200 mg kg-1 the effect of kakkalide was significant. The same dose of kakkalide prevented increased serum glutamic oxaloacetic transaminase and glutamic pyruvic transaminase activity. At a dose of 200 mg kg-1 it also counteracted ethanol-induced elevation of glucose levels. These results suggest that kakkalide might be useful for counteracting the effects of alcohol and might be effective for treating hepatic injury.

MeSH terms

  • Acute Disease
  • Animals
  • Disaccharides / therapeutic use*
  • Ethanol / toxicity
  • Glycosides*
  • Hyperglycemia / chemically induced
  • Hyperglycemia / prevention & control
  • Isoflavones / therapeutic use*
  • Liver Diseases, Alcoholic / prevention & control*
  • Male
  • Mice
  • Mice, Inbred Strains
  • Plant Extracts / therapeutic use*
  • Plants, Medicinal / chemistry*

Substances

  • Disaccharides
  • Glycosides
  • Isoflavones
  • Plant Extracts
  • Ethanol
  • kakkalide