Tumor specific contrast enhancement study of Mn-metalloporphyrin (ATN-10)--comparison of rat brain tumor model, cytotoxic and vasogenic edema models

Acta Neurochir Suppl. 1997:70:167-9. doi: 10.1007/978-3-7091-6837-0_51.

Abstract

ATN-10, Mn-metalloporphyrin, has been developed as a tumor selective contrast agent for magnetic resonance (MR) imaging. To investigate the tumor specificity of ATN-10, we produced three experimental in vivo models; rat bran tumor (9L glioma) model, vasogenic (cold injury) and cytotoxic brain edema (24-hour MCA occlusion) models. The time course of contrast enhancement was compared after intravenous injection of ATN-10 or Gd-DTPA, measuring the signal intensity of the region of interest. After ATN-10 administration, the 9L glioma model showed early (5 min) and delayed (24 hr-) peak enhancement whereas the cold injury model showed only early enhancement and the 24-hour MCA occlusion model did not show significant enhancement. After Gd-DTPA administration, all three models showed similar pattern of only early enhancement. As a contrast agent for MR imaging, ATN-10 showed different behavior than Gd-DTPA in demonstrating the blood-brain barrier disruption and moreover ATN-10 showed selective enhancement in experimental brain tumors.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Blood-Brain Barrier / physiology
  • Brain Edema / diagnosis*
  • Brain Neoplasms / diagnosis*
  • Cell Survival / physiology
  • Cold Temperature
  • Contrast Media*
  • Deuteroporphyrins*
  • Disease Models, Animal
  • Gadolinium DTPA
  • Glioma / diagnosis*
  • Indium Radioisotopes
  • Magnetic Resonance Imaging / methods*
  • Male
  • Rats
  • Rats, Inbred F344

Substances

  • Contrast Media
  • Deuteroporphyrins
  • Indium Radioisotopes
  • ATN 10
  • Gadolinium DTPA