Effect of human neutrophil elastase on tracheal mucociliary transport in anesthetized quails

Jpn J Pharmacol. 1997 Dec;75(4):439-42. doi: 10.1254/jjp.75.439.

Abstract

We investigated the effect of human neutrophil elastase (HNE) on tracheal mucociliary transport in anesthetized quails. Topical application of HNE (30-300 microg/kg) to tracheal mucosa dose-dependently decreased mucociliary transport velocity (MCTV). The HNE (300 microg/kg)-induced decrease in MCTV was blocked by ONO-5046 x Na (sodium N-[2-[4-(2,2-dimethylpropionyloxy)phenyl-sulfonylamino]benzo yl]aminoacetate tetrahydrate) (3-30 mg/kg, i.m.), a specific neutrophil elastase inhibitor. Furthermore, we found that HNE increased DNA, fucose and protein contents of tracheal lavages, and the increases were also reverted by ONO-5046 Na. These results indicated that HNE decreased tracheal mucociliary transport, and the decrease may be, at least in part, ascribed to the deterioration of tracheal secretions.

MeSH terms

  • Animals
  • Bronchoalveolar Lavage Fluid / chemistry
  • DNA / analysis
  • Dose-Response Relationship, Drug
  • Fucose / analysis
  • Glycine / analogs & derivatives*
  • Glycine / pharmacology
  • Humans
  • Leukocyte Elastase / antagonists & inhibitors
  • Leukocyte Elastase / pharmacology*
  • Male
  • Mucociliary Clearance / drug effects*
  • Mucous Membrane / drug effects
  • Mucous Membrane / metabolism
  • Proteins / analysis
  • Quail
  • Serine Proteinase Inhibitors / pharmacology*
  • Sulfonamides / pharmacology*
  • Trachea / drug effects*
  • Trachea / metabolism

Substances

  • Proteins
  • Serine Proteinase Inhibitors
  • Sulfonamides
  • Fucose
  • DNA
  • sivelestat
  • Leukocyte Elastase
  • Glycine