Applicability of the free energies of solvation for the prediction of ecotoxicity: study of chlorophenols

SAR QSAR Environ Res. 1997;6(3-4):163-81. doi: 10.1080/10629369708033250.

Abstract

Free energies of solvation of chlorophenols were calculated in two solvents: water and n-hexadecane from the AMSOL program. These free energies of solvation are the sum of two terms: polarization free energies (delta GENP) and cavity, dispersion, solvent structure free energies (G degree CDS). This study shows, in the case of chlorophenols, that a direct relation exists between one of the two components for the calculation of free energy (G degree CDS) in water and n-hexadecane, and the ecotoxicity values for five biological systems. We point out the interest of using these new descriptors in QSAR study.

MeSH terms

  • Chlorophenols / chemistry*
  • Chlorophenols / toxicity*
  • Ecosystem
  • Molecular Conformation
  • Predictive Value of Tests
  • Solutions
  • Structure-Activity Relationship
  • Thermodynamics
  • Water Pollutants, Chemical / toxicity*

Substances

  • Chlorophenols
  • Solutions
  • Water Pollutants, Chemical