Phospholipase D hydrolyzes short-chain analogs of phosphatidylcholine in the absence of detergent

Lipids. 1998 Feb;33(2):223-7. doi: 10.1007/s11745-998-0199-5.

Abstract

Phospholipase D is an important enzyme in signal transduction in neuronal tissue. A variety of assays have been used to measure phospholipase D activity in vitro. The most typical measure of phospholipase D activity is the production of phosphatidylethanol in the presence of ethanol. Phosphatidylethanol is a product of transphosphatidylation activity that is considered a unique property of phospholipase D. To support transphosphatidylation activity, high concentrations of ethanol may be required. Furthermore, most assays in the literature utilize a detergent. These extreme conditions, detergent and ethanol, may alter phospholipase D and hinder the study of its regulation. In this manuscript we describe an assay that eliminates these potentially confounding conditions. It utilizes high specific activity [3H]butanol as a nucleophilic receptor. This eliminates the need for high concentrations of alcohol. The substrate is an analog of phosphatidylcholine that contains short-chain fatty acids, 1,2-dioctanoyl-sn-glycero-3-phosphocholine. Phospholipase D readily hydrolyzes this substrate in the absence of detergent. This novel assay should be useful in the further characterization of phospholipase D.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Animals
  • Brain / enzymology
  • Butanols / metabolism
  • Detergents
  • Hydrolysis
  • Microsomes / enzymology
  • Nerve Tissue Proteins / metabolism*
  • Phosphatidylcholines / metabolism*
  • Phospholipase D / metabolism*
  • Rats

Substances

  • 1,2-dioctanoyl-sn-glycero-3-phosphocholine
  • Butanols
  • Detergents
  • Nerve Tissue Proteins
  • Phosphatidylcholines
  • Phospholipase D