Absence of cross-reactivity of SR90107A/ORG31540 pentasaccharide with antibodies to heparin-PF4 complexes developed in heparin-induced thrombocytopenia

Blood Coagul Fibrinolysis. 1997 Mar;8(2):114-7. doi: 10.1097/00001721-199703000-00005.

Abstract

New carbohydrate-based anticoagulants devoid of the side effects of unfractionated heparin are currently under development and show a major potential for patients with heparin-induced thrombocytopenia (HIT) who still require efficient antithrombotic therapy. As HIT is usually associated with antibodies to heparin-platelet factor 4 (H-PF4) complexes, cross-reactivity of the heparin pentasaccharide SR90107A/ORG31540 was tested in the presence of PF4 with the plasma from 49 patients with HIT. No cross-reactivity was observed whatever the pentasaccharide concentrations. Although more extensive studies are required for excluding its total absence of immunogenicity and pathogenicity, this pentasaccharide is a candidate for use in emergency situations in patients with HIT.

Publication types

  • Clinical Trial

MeSH terms

  • Autoantibodies / immunology*
  • Cross Reactions
  • Enzyme-Linked Immunosorbent Assay
  • Female
  • Fibrinolytic Agents / immunology*
  • Fibrinolytic Agents / therapeutic use
  • Heparin / adverse effects*
  • Heparin / immunology
  • Humans
  • Macromolecular Substances
  • Male
  • Oligosaccharides / immunology*
  • Oligosaccharides / therapeutic use
  • Platelet Factor 4 / immunology*
  • Postoperative Care
  • Thrombocytopenia / chemically induced*
  • Thrombocytopenia / immunology*
  • Thrombosis / drug therapy

Substances

  • Autoantibodies
  • Fibrinolytic Agents
  • Macromolecular Substances
  • Oligosaccharides
  • PENTA
  • Platelet Factor 4
  • Heparin