Occupational contact dermatitis to propacetamol. Allergological and chemical investigations in two new cases

Dermatology. 1997;195(4):329-31. doi: 10.1159/000245982.

Abstract

Background and objective: In 2 new cases of occupational contact dermatitis due to a recently described allergen (propacetamol), a prodrug which is a soluble diethylglycidyl ester of paracetamol, an allergological investigation was performed to elucidate the nature of the allergen involved in the propacetamol contact sensitivity.

Observations: Two nurses with eczema of the hands and face had positive patch tests to Pro-Dafalgan. Every day the nurses prepared injections of Pro-Dafalgan (propacetamol dissolved in sodium citrate). The sensitization was due to propacetamol and not to the solvent. To elucidate which part of propacetamol was responsible for the sensitization, the 2 nurses were patch-tested with diethylamine, paracetamol (diluted in different vehicles) and some of their chemical analogues and potential impurities which were all negative.

Conclusions: Propacetamol induces airborne contact dermatitis with no evidence of sensitization to paracetamol or diethylglycine, possibly because of either the presence of unknown impurities and/or an antigenic structure related to the covalent bond of the prodrug.

Publication types

  • Case Reports

MeSH terms

  • Acetaminophen / adverse effects
  • Acetaminophen / analogs & derivatives*
  • Acetaminophen / chemistry
  • Acetaminophen / immunology
  • Adult
  • Allergens / immunology
  • Analgesics / adverse effects*
  • Analgesics / chemistry
  • Analgesics / immunology
  • Anti-Inflammatory Agents, Non-Steroidal / adverse effects*
  • Anti-Inflammatory Agents, Non-Steroidal / chemistry
  • Anti-Inflammatory Agents, Non-Steroidal / immunology
  • Antigens / immunology
  • Dermatitis, Occupational / etiology*
  • Diethylamines / adverse effects
  • Diethylamines / immunology
  • Drug Contamination
  • Eczema / chemically induced
  • Facial Dermatoses / chemically induced
  • Hand Dermatoses / chemically induced
  • Humans
  • Immunization
  • Nurses
  • Patch Tests
  • Pharmaceutical Vehicles
  • Prodrugs / adverse effects*
  • Prodrugs / chemistry

Substances

  • Allergens
  • Analgesics
  • Anti-Inflammatory Agents, Non-Steroidal
  • Antigens
  • Diethylamines
  • Pharmaceutical Vehicles
  • Prodrugs
  • Acetaminophen
  • propacetamol
  • diethylamine