Therapeutic effects of an injectable new quinolone, pazufloxacin, against polymicrobial infections in the uterine endometritis model

Chemotherapy. 1998 Mar-Apr;44(2):99-102. doi: 10.1159/000007099.

Abstract

Polymicrobial infections with aerobes and anaerobes are common in female genital tract infections. We evaluated the efficacy of an injectable new quinolon, pazufloxacin, using a uterine endometritis model. Rats were infected with a mixed inoculation of Escherichia coli plus Bacteriodes fragilis (MIC of pazufloxacin and ceftazidime: E. coli: 0.05 and 1.56 micrograms/ml, respectively, B. fragilis: 3.13 and 3.13 micrograms/ml, respectively). After inoculating 10(7) cfu/rat of each organism, pazufloxacin or ceftazidime (10 or 20 mg/kg, respectively, i.v., b.i.d., 3 days) was administered and compared with the nontreated group. The viable cell counts of the uterine corpus and uterine cervix in pazufloxacin-treated and ceftazidime-treated groups were decreased, compared with the nontreated group. The viable cell counts of the adnexa in the pazufloxacin-treated group were significantly decreased, compared with the ceftazidimetreated group. These results suggest that pazufloxacin would be useful for the treatment of polymicrobial infections, especially adnexitis.

Publication types

  • Comparative Study

MeSH terms

  • Animals
  • Anti-Infective Agents / administration & dosage
  • Anti-Infective Agents / therapeutic use*
  • Bacteroides Infections*
  • Bacteroides fragilis / drug effects*
  • Ceftazidime / administration & dosage
  • Ceftazidime / therapeutic use
  • Cephalosporins / administration & dosage
  • Cephalosporins / therapeutic use
  • Colony Count, Microbial
  • Disease Models, Animal
  • Dose-Response Relationship, Drug
  • Endometritis / drug therapy*
  • Endometritis / microbiology*
  • Escherichia coli Infections*
  • Female
  • Fluoroquinolones*
  • Genital Diseases, Female / drug therapy
  • Genital Diseases, Female / microbiology
  • Injections, Intravenous
  • Microbial Sensitivity Tests
  • Oxazines / administration & dosage
  • Oxazines / therapeutic use*
  • Rats
  • Rats, Sprague-Dawley
  • Species Specificity

Substances

  • Anti-Infective Agents
  • Cephalosporins
  • Fluoroquinolones
  • Oxazines
  • pazufloxacin
  • Ceftazidime