Effect of endoplasmic Ca2+-ATPase inhibitors on cochlear potentials in the guinea-pig

Acta Otolaryngol. 1998 Mar;118(2):198-205. doi: 10.1080/00016489850154900.

Abstract

The effect of endoplasmic Ca2+-ATPase inhibitors on cochlear potentials was examined in the guinea-pig. Perilymphatic perfusion with thapsigargin (10[-6] M) produced a significant decrease in the amplitudes of cochlear microphonics, negative summating potential and compound action potential, and a significant prolongation of N1 latency with no change in the endocochlear potential. These changes were all dose dependent. Another endoplasmic Ca2+-ATPase inhibitor, cyclopiazonic acid (10[-5] M), produced the same effects as thapsigargin on cochlear potentials. These results suggest that endoplasmic Ca2+-ATPase inhibitors may have inhibitory functions on cochlear potentials.

MeSH terms

  • Animals
  • Calcium-Transporting ATPases / antagonists & inhibitors*
  • Cochlea / drug effects*
  • Cochlea / physiology
  • Dose-Response Relationship, Drug
  • Enzyme Inhibitors / pharmacology
  • Guinea Pigs
  • Indoles / pharmacology
  • Membrane Potentials / drug effects
  • Thapsigargin / pharmacology

Substances

  • Enzyme Inhibitors
  • Indoles
  • Thapsigargin
  • Calcium-Transporting ATPases
  • cyclopiazonic acid