The determination of pamidronate in pharmaceutical preparations by ion-pair liquid chromatography after derivatization with phenylisothiocyanate

J Pharm Biomed Anal. 1997 Nov;16(3):491-7. doi: 10.1016/s0731-7085(97)00090-3.

Abstract

An analytical method was developed for the determination of pamidronate [(3-amino-1-hydroxypropylidene)bisphosphonate] by ion-pair liquid chromatography. The analyte was derivatized with phenylisothiocyanate into an UV-absorbing derivative. The reaction product was cleaned-up by a double ion-pair extraction and treated with hydrogen peroxide prior to injection. Both, the detection limit and the lower limit of quantification of pamidronate in water were 0.1 microgram ml-1 disodium pamidronate. The intra-day precision was 3% for a 5-microgram ml-1 pamidronate standard solution and the inter-day precision 6% for a 3-microgram ml-1 solution. The method was applied in the quality control of pamidronate injection concentrates and tablets.

MeSH terms

  • Chromatography, High Pressure Liquid
  • Chromatography, Liquid
  • Diphosphonates / analysis*
  • Indicators and Reagents
  • Isothiocyanates
  • Pamidronate
  • Thiocyanates

Substances

  • Diphosphonates
  • Indicators and Reagents
  • Isothiocyanates
  • Thiocyanates
  • phenylisothiocyanate
  • Pamidronate