Serotonin3 receptor antagonism of alcohol intake: effects of drinking conditions

Alcohol. 1998 May;15(4):291-8. doi: 10.1016/s0741-8329(97)00132-8.

Abstract

The effects of 5-HT3 receptor antagonists on ethanol intake were examined in the selectively bred alcohol-preferring P line of rats under continuous and limited access to 10% (v/v) ethanol with food and water ad lib. Single daily injections of either MDL 72222 (MDL) or ICS 205-930 (ICS) (0.01-3.0 mg/kg, SC) given 60 min before a 4-h scheduled access period for 4 consecutive days failed at all doses to alter the intake of a 10% (v/v) ethanol solution by P rats. However, multiple daily injections of either MDL (1-3 mg/kg, SC) or ICS (3.0 and 5.0 mg/kg, SC), given three times daily at 4-h intervals, significantly reduced ethanol intake under 24-h free-choice conditions on the first treatment day. Additionally, a single administration of 1.0 mg/kg MDL reduced 24-h free-choice ethanol intake by approximately 50% of control values and had no effect on 24-h saccharin intake. The effects of MDL were further examined in a 2-h schedule access paradigm in which rats received the access period at the same time every day (Fixed) or randomly during the dark cycle (Variable). Although 1.0 mg/kg MDL had little effect on ethanol drinking in the Fixed group, ethanol intake was reduced by 55% of control levels in the Variable group. Overall, the data indicate that drinking conditions influence the effectiveness of 5-HT3 antagonists to reduce ethanol consumption. Furthermore, the results suggest that conditions, associated with limited access ethanol drinking, markedly reduce the actions of 5-HT3 antagonists on ethanol intake.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Alcohol Drinking / physiopathology*
  • Animals
  • Drinking / drug effects
  • Drug Administration Schedule
  • Female
  • Indoles / administration & dosage*
  • Indoles / pharmacology
  • Injections, Subcutaneous
  • Rats
  • Rats, Inbred Strains
  • Saccharin
  • Serotonin Antagonists / administration & dosage*
  • Serotonin Antagonists / pharmacology
  • Solutions
  • Tropanes / administration & dosage*
  • Tropanes / pharmacology
  • Tropisetron

Substances

  • Indoles
  • Serotonin Antagonists
  • Solutions
  • Tropanes
  • Tropisetron
  • Saccharin
  • bemesetron