Central CRF inhibits gastric emptying of a nutrient solid meal in rats: the role of CRF2 receptors

Am J Physiol. 1998 May;274(5):G965-70. doi: 10.1152/ajpgi.1998.274.5.G965.

Abstract

Corticotropin-releasing factor (CRF)-related peptides exhibit different affinity for the receptor subtypes 1 and 2 cloned in the rat brain. We investigated, in conscious rats, the effects of intracisternal (i.c.) injection of CRF (rat/human) on the 5-h rate of gastric emptying of a solid nutrient meal (Purina chow and water ad libitum for 3 h) and the CRF receptor subtype involved. CRF, urotensin I (suckerfish), and sauvagine (frog) injected i.c. inhibited gastric emptying in a dose-dependent manner, with ED50 values of 0.31, 0.13, and 0.08 microgram/rat, respectively. Rat CRF-(6-33) (0.1-10 micrograms i.c.) had no effect. The nonselective CRF1 and CRF2 receptor antagonist, astressin, injected i.c. completely blocked the inhibitory effect of i.c. CRF, urotensin I, and sauvagine with antagonist-to-agonist ratios of 3:1, 10:1, and 16:1, respectively. The CRF1-selective receptor antagonist NBI-27914 injected i.c. at a ratio of 170:1 had no effect. These data show that central CRF and CRF-related peptides are potent inhibitors of gastric emptying of a solid meal with a rank order of potency characteristic of the CRF2 receptor subtype affinity (sauvagine > urotensin I > CRF). In addition, the reversal by astressin but not by the CRF1-selective receptor antagonist further supports the view that the CRF2 receptor subtype is primarily involved in central CRF-induced delayed gastric emptying.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Amphibian Proteins
  • Animal Feed*
  • Animals
  • Brain / physiology*
  • Corticotropin-Releasing Hormone / antagonists & inhibitors
  • Corticotropin-Releasing Hormone / pharmacology*
  • Gastric Emptying / drug effects*
  • Injections, Intraventricular
  • Male
  • Peptide Fragments / pharmacology
  • Peptide Hormones
  • Peptides / antagonists & inhibitors
  • Peptides / pharmacology
  • Rats
  • Rats, Sprague-Dawley
  • Receptors, Corticotropin-Releasing Hormone / physiology*
  • Urotensins / antagonists & inhibitors
  • Urotensins / pharmacology

Substances

  • Amphibian Proteins
  • Peptide Fragments
  • Peptide Hormones
  • Peptides
  • Receptors, Corticotropin-Releasing Hormone
  • Urotensins
  • astressin
  • sauvagine
  • Corticotropin-Releasing Hormone
  • urotensin I