Molecular cloning of xSRC-3, a novel transcription coactivator from Xenopus, that is related to AIB1, p/CIP, and TIF2

Mol Endocrinol. 1998 Jul;12(7):1038-47. doi: 10.1210/mend.12.7.0139.

Abstract

Nuclear receptors regulate transcription by binding to specific DNA response elements of target genes. Herein, we report the molecular cloning and characterization of a novel Xenopus cDNA encoding a transcription coactivator xSRC-3 by using retinoid X receptor (RXR) as a bait in the yeast two-hybrid screening. It belongs to a growing coactivator family that includes a steroid receptor coactivator amplified in breast cancer (AIB1), p300/ CREB-binding protein (CBP)-interacting protein (p/ CIP), and transcriptional intermediate factor 2 (TIF2). It also interacts with a series of nuclear receptors including retinoic acid receptor (RAR), thyroid hormone receptor (TR), and orphan nuclear receptors [hepatocyte nuclear receptor 4 (HNF4) and constitutive androstane receptor (CAR)]. However, it does not interact with small heterodimer partner (SHP), an orphan nuclear receptor known to antagonize ligand-dependent transactivation of other nuclear receptors. In CV-1 cells, cotransfection of xSRC-3 differentially stimulates ligand-induced transactivation of RXR, TR, and RAR in a dose-dependent manner. Interestingly, xSRC-3 is highly expressed in adult liver and early stages of oocyte development, suggesting that studies of xSRC-3 may lead to better understanding of the roles nuclear receptors play in oocyte development as well as liver-specific gene expression.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetyltransferases
  • Alternative Splicing
  • Amino Acid Sequence
  • Animals
  • Binding Sites
  • Cell Nucleus / metabolism
  • Cloning, Molecular*
  • Female
  • Gene Expression
  • Histone Acetyltransferases
  • Humans
  • Molecular Sequence Data
  • Mutagenesis
  • Nuclear Receptor Coactivator 1
  • Nuclear Receptor Coactivator 2
  • Nuclear Receptor Coactivator 3
  • Oncogene Proteins
  • Receptors, Retinoic Acid / metabolism
  • Receptors, Thyroid Hormone / metabolism
  • Recombinant Fusion Proteins
  • Retinoid X Receptors
  • Saccharomyces cerevisiae / genetics
  • Sequence Homology
  • Trans-Activators* / chemistry
  • Trans-Activators* / genetics*
  • Trans-Activators* / metabolism
  • Transcription Factors* / chemistry
  • Transcription Factors* / metabolism
  • Transcriptional Activation
  • Xenopus Proteins*
  • Xenopus*

Substances

  • NCOA2 protein, human
  • NCOA3 protein, Xenopus
  • Nuclear Receptor Coactivator 2
  • Oncogene Proteins
  • Receptors, Retinoic Acid
  • Receptors, Thyroid Hormone
  • Recombinant Fusion Proteins
  • Retinoid X Receptors
  • Trans-Activators
  • Transcription Factors
  • Xenopus Proteins
  • Acetyltransferases
  • Histone Acetyltransferases
  • NCOA1 protein, human
  • NCOA3 protein, human
  • Nuclear Receptor Coactivator 1
  • Nuclear Receptor Coactivator 3