Radioprotection of salivary glands by amifostine in high-dose radioiodine therapy

J Nucl Med. 1998 Jul;39(7):1237-42.

Abstract

Salivary gland impairment after high-dose radioiodine treatment is well recognized. Because differentiated thyroid cancer has a good prognosis, reduction of long-term side effects is important. This study investigated the radioprotective effects of amifostine in animals and humans receiving high-dose radioiodine therapy.

Methods: Quantitative salivary gland scintigraphy was performed in five rabbits before and up to 3 mo after high-dose radioiodine therapy applying 1 GBq 131I. Three animals received 200 mg/kg amifostine before high-dose radioiodine therapy, and two served as controls. All animals were examined histopathologically. Quantitative salivary gland scintigraphy also was performed in 17 patients with differentiated thyroid cancer before and 3 mo after high-dose radioiodine therapy with 6 GBq 131I. Eight patients were treated with 500 mg/m2 amifostine before high-dose radioiodine therapy, and nine served as controls.

Results: In two control rabbits, high-dose radioiodine therapy significantly reduced parenchymal function by 63% and 46% in parotid and submandibular glands, respectively. In contrast, there was no significant decrease in parenchymal function in amifostine-treated animals. Histopathologically, lipomatosis was observed in control animals but was negligible in amifostine-treated animals. Similar findings were observed in differentiated thyroid cancer patients. In nine control patients, high-dose radioiodine therapy significantly (p < 0.01) reduced parenchymal function by 37% and 31% in parotid and submandibular glands, respectively. Three patients exhibited Grade I (World Health Organization) xerostomia. In contrast, there was no significant decrease in parenchymal function in amifostine-treated patients and no incidence of xerostomia.

Conclusion: Parenchymal damage in salivary glands induced by high-dose radioiodine therapy can be reduced significantly by amifostine. This may increase the quality of life of patients with differentiated thyroid cancer.

MeSH terms

  • Adenocarcinoma, Follicular / radiotherapy
  • Adult
  • Aged
  • Amifostine / therapeutic use*
  • Animals
  • Carcinoma, Papillary / radiotherapy
  • Case-Control Studies
  • Female
  • Humans
  • Iodine Radioisotopes / administration & dosage*
  • Male
  • Middle Aged
  • Rabbits
  • Radiation-Protective Agents / therapeutic use*
  • Radionuclide Imaging
  • Radiotherapy Dosage
  • Salivary Glands / diagnostic imaging
  • Salivary Glands / radiation effects*
  • Sodium Pertechnetate Tc 99m
  • Thyroid Neoplasms / radiotherapy*

Substances

  • Iodine Radioisotopes
  • Radiation-Protective Agents
  • Sodium Pertechnetate Tc 99m
  • Amifostine