Stability of mycophenolate mofetil as an extemporaneous suspension

Ann Pharmacother. 1998 Jul-Aug;32(7-8):755-7. doi: 10.1345/aph.17213.

Abstract

Objective: To evaluate the physical and chemical stability of a suspension of mycophenolate mofetil (MMF) prepared in the hospital from commercially available MMF capsules.

Methods: Suspensions of MMF were prepared at room temperature and stored at 5, 25, 37, and 45 degrees C over a period of 50 to 210 days. The contents of MMF and its degradation product, mycophenolic acid, in the suspension were measured at various time points by HPLC.

Results: MMF suspensions were stable (as determined by the presence of > or = 90% of the labeled amount) at 45 degrees C for at least 11 days, at 37 degrees C for at least 28 days, at 25 degrees C for at least 28 days, and at 5 degrees C for at least 210 days. The suspension was also physically stable at 5 degrees C during the entire test period.

Conclusions: The compounded MMF suspension was stable for at least 11 days at all the temperatures studied and for as long as 210 days at 5 degrees C. This formulation appears to be clinically acceptable and provides a convenient dosage form for pediatric patients and for adults during the early postoperative period.

MeSH terms

  • Chromatography, High Pressure Liquid
  • Drug Stability
  • Humans
  • Immunosuppressive Agents / chemistry*
  • Middle Aged
  • Mycophenolic Acid / analogs & derivatives*
  • Mycophenolic Acid / chemistry
  • Suspensions / analysis
  • Suspensions / chemistry
  • Temperature
  • Time Factors

Substances

  • Immunosuppressive Agents
  • Suspensions
  • Mycophenolic Acid