In vitro activity of loracarbef against TEM extended-spectrum beta-lactamase-producing Escherichia coli strains and its interaction with the enzymes

Chemotherapy. 1998 Jul-Aug;44(4):260-4. doi: 10.1159/000007122.

Abstract

The in vitro activity of loracarbef was evaluated against Escherichia coli strains producing TEM extended-spectrum beta-lactamases (ESBLs). The MICs of loracarbef were lower than those of cefaclor and cephalothin. The antibiotic was active (MICs < or = 2 mg/l) against strains producing TEM-6, TEM-8, TEM-10, TEM-16, TEM-26 and TEM-28 beta-lactamases. The MICs for TEM-3-, TEM-5- and TEM-24-producing strains were higher (> or = 16 mg/l). Hydrolysis studies indicated that the latter beta-lactamases inactivated loracarbef more efficiently than the remaining TEM-type ESBLs examined.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cephalosporins / metabolism
  • Cephalosporins / pharmacology*
  • Drug Stability
  • Escherichia coli / drug effects*
  • Escherichia coli / enzymology
  • Hydrolysis
  • Microbial Sensitivity Tests
  • Plasmids / genetics
  • beta-Lactam Resistance
  • beta-Lactamases / chemistry
  • beta-Lactamases / metabolism*

Substances

  • Cephalosporins
  • loracarbef
  • beta-Lactamases