Effect of Ca2+ and cAMP on capacitance-measured hormone secretion in human GH-secreting adenoma cells

Am J Physiol. 1998 Oct;275(4):E649-54. doi: 10.1152/ajpendo.1998.275.4.E649.

Abstract

Membrane capacitance (Cm) was measured as an index of exocytosis in human growth hormone-secreting adenoma cells using the perforated whole cell, patch-clamp technique; the effects of membrane depolarization, growth hormone-releasing hormone, and 8-bromoadenosine 3',5'-cyclic monophosphate (8-BrcAMP) were examined. Cm was increased by membrane depolarization to potentials beyond the threshold necessary to open voltage-gated Ca2+ channels. These voltage-dependent changes in Cm varied as a function of both depolarization amplitude and duration and were blocked in the presence of the Ca2+ channel antagonist nitrendipine (10(-6) M). When membrane potential was clamped at the holding potential (-78 mV), voltage-gated Ca2+ channels were closed, and neither application of growth hormone-releasing hormone nor 8-BrcAMP affected Cm. However, when these agents were applied to depolarized cells, where the voltage-gated Ca2+ channels were open, the increases in Cm were augmented. From these data, it was concluded that elevation of intracellular cAMP, per se, did not stimulate exocytosis. Rather, Ca2+ influx through voltage-gated channels was a prerequisite for cAMP-induced exocytosis.

MeSH terms

  • 8-Bromo Cyclic Adenosine Monophosphate / pharmacology
  • Adenoma / metabolism*
  • Adenoma / physiopathology*
  • Calcium / physiology*
  • Calcium Channels / physiology
  • Cyclic AMP / physiology*
  • Exocytosis / drug effects
  • Exocytosis / physiology
  • Human Growth Hormone / metabolism*
  • Humans
  • Ion Channel Gating / drug effects
  • Ion Channel Gating / physiology
  • Membrane Potentials / drug effects
  • Membrane Potentials / physiology
  • Nitrendipine / pharmacology
  • Patch-Clamp Techniques
  • Pituitary Neoplasms / metabolism*
  • Pituitary Neoplasms / physiopathology*
  • Tumor Cells, Cultured

Substances

  • Calcium Channels
  • Human Growth Hormone
  • 8-Bromo Cyclic Adenosine Monophosphate
  • Nitrendipine
  • Cyclic AMP
  • Calcium