An essential lysine residue of green crab (Scylla Serrata) alkaline phosphatase

Biochem Mol Biol Int. 1998 Oct;46(2):225-31. doi: 10.1080/15216549800203732.

Abstract

The values of pKa (10.38) and Hion (10.92 Kcal/mol) have been determined for the ionizing groups controlling activity of green crab alkaline phosphatase. The results suggest that -NH2 of lysine residue responsible for the ionization with pKc = 10.38 and delta H(o)ion = 10.92 Kcal/mol is in the active site of the enzyme. Modification of lysine residues of the enzyme by an excess of 2,4,6-trinitrobenzenesulfonic acid leads to complete inactivation. The two results coincide with each other. Quantitative assessment of the data indicates that among the reactive -NH2 groups modified only one is essential for the activity of the enzyme.

MeSH terms

  • Alkaline Phosphatase / antagonists & inhibitors
  • Alkaline Phosphatase / chemistry
  • Alkaline Phosphatase / metabolism*
  • Animals
  • Binding Sites
  • Brachyura / enzymology*
  • Dose-Response Relationship, Drug
  • Enzyme Inhibitors / pharmacology
  • Hydrogen-Ion Concentration
  • Kinetics
  • Lysine / metabolism*
  • Temperature
  • Thermodynamics
  • Trinitrobenzenesulfonic Acid / pharmacology

Substances

  • Enzyme Inhibitors
  • Trinitrobenzenesulfonic Acid
  • Alkaline Phosphatase
  • Lysine