Inhibition of beta-catenin-mediated transactivation by cadherin derivatives

Proc Natl Acad Sci U S A. 1998 Dec 22;95(26):15339-44. doi: 10.1073/pnas.95.26.15339.

Abstract

We studied the effect of N-cadherin, and its free or membrane-anchored cytoplasmic domain, on the level and localization of beta-catenin and on its ability to induce lymphocyte enhancer-binding factor 1 (LEF-1)-responsive transactivation. These cadherin derivatives formed complexes with beta-catenin and protected it from degradation. N-cadherin directed beta-catenin into adherens junctions, and the chimeric protein induced diffuse distribution of beta-catenin along the membrane whereas the cytoplasmic domain of N-cadherin colocalized with beta-catenin in the nucleus. Cotransfection of beta-catenin and LEF-1 into Chinese hamster ovary cells induced transactivation of a LEF-1 reporter, which was blocked by the N-cadherin-derived molecules. Expression of N-cadherin and an interleukin 2 receptor/cadherin chimera in SW480 cells relocated beta-catenin from the nucleus to the plasma membrane and reduced transactivation. The cytoplasmic tails of N- or E-cadherin colocalized with beta-catenin in the nucleus, and suppressed the constitutive LEF-1-mediated transactivation, by blocking beta-catenin-LEF-1 interaction. Moreover, the 72 C-terminal amino acids of N-cadherin stabilized beta-catenin and reduced its transactivation potential. These results indicate that beta-catenin binding to the cadherin cytoplasmic tail either in the membrane, or in the nucleus, can inhibit beta-catenin degradation and efficiently block its transactivation capacity.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • CHO Cells
  • Cadherins / chemistry
  • Cadherins / physiology*
  • Cell Line
  • Cell Membrane / metabolism
  • Cell Nucleus / metabolism
  • Chickens
  • Cricetinae
  • Cytoskeletal Proteins / genetics
  • Cytoskeletal Proteins / physiology*
  • DNA-Binding Proteins / metabolism*
  • Kinetics
  • Lymphoid Enhancer-Binding Factor 1
  • Plasmids
  • Receptors, Interleukin-2 / genetics
  • Receptors, Interleukin-2 / physiology*
  • Recombinant Fusion Proteins / metabolism
  • Trans-Activators*
  • Transcription Factors / metabolism*
  • Transcriptional Activation*
  • Transfection
  • beta Catenin

Substances

  • Cadherins
  • Cytoskeletal Proteins
  • DNA-Binding Proteins
  • Lymphoid Enhancer-Binding Factor 1
  • Receptors, Interleukin-2
  • Recombinant Fusion Proteins
  • Trans-Activators
  • Transcription Factors
  • beta Catenin