Novel euglycemic and hypolipidemic agents: Part-2. Antioxidant moiety as structural motif

Bioorg Med Chem Lett. 1998 May 5;8(9):999-1002. doi: 10.1016/s0960-894x(98)00159-0.

Abstract

Several thiazolidinediones having antioxidant moities in their structural motif have been synthesised and evaluated for their euglycemic and hypolipidemic activities. A few of them have been found to be superior to troglitazone.

MeSH terms

  • Animals
  • Antioxidants / chemical synthesis*
  • Antioxidants / chemistry
  • Antioxidants / pharmacology
  • Blood Glucose / metabolism
  • Diabetes Mellitus, Type 2 / blood
  • Diabetes Mellitus, Type 2 / drug therapy
  • Diabetes Mellitus, Type 2 / genetics
  • Drug Design
  • Hypoglycemic Agents / chemical synthesis*
  • Hypoglycemic Agents / chemistry
  • Hypoglycemic Agents / pharmacology
  • Hypolipidemic Agents / chemical synthesis*
  • Hypolipidemic Agents / chemistry
  • Hypolipidemic Agents / pharmacology
  • Indicators and Reagents
  • Mice
  • Mice, Mutant Strains
  • Structure-Activity Relationship
  • Thiazoles / chemical synthesis*
  • Thiazoles / chemistry
  • Thiazoles / pharmacology
  • Triglycerides / blood

Substances

  • Antioxidants
  • Blood Glucose
  • Hypoglycemic Agents
  • Hypolipidemic Agents
  • Indicators and Reagents
  • Thiazoles
  • Triglycerides