Effect of gemfibrozil on serum levels of prostacyclin and precursor fatty acids in hyperlipidemic patients with Type 2 diabetes

Diabetes Res Clin Pract. 1998 Dec;42(3):149-54. doi: 10.1016/s0168-8227(98)00107-7.

Abstract

Lipid-lowering fibrate drugs are known to affect the synthesis of fatty acids, which may alter the prostacyclin synthesis in diabetic patients. Therefore, the serum levels of precursor fatty acids and 6-keto-prostaglandin F1alpha (6-keto PGF1alpha) were determined in ten hyperlipidemic patients with Type 2 diabetes before and after administration of gemfibrozil (900 mg/day) for 3 months, in comparison with the results in seven non-diabetic hyperlipidemic patients. Gemfibrozil significantly reduced the serum concentration of dihomo-7-linolenic acid, total cholesterol and triglycerides, but did not affect the serum levels of arachidonic acid and 6-keto PGF1alpha in diabetic and non-diabetic patients. Thus, gemfibrozil did not affect the synthesis of prostacyclin in spite of the reduction of precursor fatty acids in diabetic and non-diabetic patients.

MeSH terms

  • 6-Ketoprostaglandin F1 alpha / blood*
  • 8,11,14-Eicosatrienoic Acid / blood
  • Aged
  • Arachidonic Acid / blood
  • Cholesterol / blood
  • Diabetes Mellitus, Type 2 / blood*
  • Diabetes Mellitus, Type 2 / complications
  • Fatty Acids, Nonesterified / blood*
  • Fatty Acids, Unsaturated / blood*
  • Female
  • Gemfibrozil / therapeutic use*
  • Humans
  • Hyperlipidemias / blood*
  • Hyperlipidemias / complications
  • Hyperlipidemias / drug therapy*
  • Hypolipidemic Agents / therapeutic use*
  • Male
  • Middle Aged
  • Time Factors
  • Triglycerides / blood

Substances

  • Fatty Acids, Nonesterified
  • Fatty Acids, Unsaturated
  • Hypolipidemic Agents
  • Triglycerides
  • Arachidonic Acid
  • 6-Ketoprostaglandin F1 alpha
  • Cholesterol
  • 8,11,14-Eicosatrienoic Acid
  • Gemfibrozil