Propanil affects transcriptional and posttranscriptional regulation of IL-2 expression in activated EL-4 cells

Toxicol Appl Pharmacol. 1999 Jan 15;154(2):153-9. doi: 10.1006/taap.1998.8545.

Abstract

The amide-class herbicide, propanil, causes numerous immunomodulary effects in animal models. In the present study, we investigated the effect of propanil on IL-2 expression and production in the murine lymphoma T cell line, EL-4. When supernatants of cells stimulated with phorbol 12-myristate 13-acetate in the presence of propanil were assessed by enzyme-linked immunosorbent assay, IL-2 levels were dose-dependently decreased by 20 and 50 microM of propanil but not at 10 microM. Quantitative Northern blot analysis of peak IL-2 message levels also showed a dose-dependent decrease. The kinetic pattern of message production, however, was unaffected. To determine if the reduced message production was due to reduced signaling or message stability, nuclear run-on and mRNA stability assays were performed. Nuclear run-on assays determined that the transcription rate of the IL-2 gene was decreased approximately 50% in the presence of 20 microM propanil, indicating that it was able to interfere with signal transduction. IL-2 message stability assays also demonstrated a reduction in message stability. Thus, propanil appears to reduce IL-2 production by affecting the signal transduction pathway and IL-2 message stability.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Carcinogens / pharmacology
  • Cell Line
  • Cell Nucleus / drug effects
  • Cell Nucleus / metabolism
  • DNA Probes
  • Herbicides / toxicity*
  • Interleukin-2 / biosynthesis*
  • Interleukin-2 / genetics
  • Propanil / toxicity*
  • Protein Processing, Post-Translational / drug effects*
  • RNA / biosynthesis
  • RNA / isolation & purification
  • Signal Transduction / drug effects
  • Tetradecanoylphorbol Acetate / pharmacology
  • Transcription, Genetic / drug effects*

Substances

  • Carcinogens
  • DNA Probes
  • Herbicides
  • Interleukin-2
  • RNA
  • Propanil
  • Tetradecanoylphorbol Acetate