Cannabimimetic activity in rats and pigeons of HU 210, a potent antiemetic drug

Pharmacol Biochem Behav. 1999 Jan;62(1):75-80. doi: 10.1016/s0091-3057(98)00114-2.

Abstract

Preliminary behavioral experiments in rats with the cannabinoid agonist HU 210 (12.5-100 microg/kg i.p.) showed that it has a potent cannabimimetic profile similar to that of delta9THC; the drug dose dependently depressed locomotor activity, rearing, and grooming and elicited vocalization and circling at the highest doses. In subsequent studies on pigeons, HU 210 (12.5-50 microg/kg s.c.) confirmed its sedative effects; it also afforded protection against vomiting induced by cisplatin (7.5 mg/kg i.v.) and emetine (20 mg/kg s.c.) and emetine-induced head shake.

MeSH terms

  • Animals
  • Antiemetics / pharmacology*
  • Columbidae
  • Dose-Response Relationship, Drug
  • Dronabinol / analogs & derivatives*
  • Dronabinol / pharmacology
  • Female
  • Grooming / drug effects
  • Hypnotics and Sedatives / pharmacology
  • Male
  • Motor Activity / drug effects
  • Rats

Substances

  • Antiemetics
  • Hypnotics and Sedatives
  • Dronabinol
  • HU 211