Activation of the signal transducer glycoprotein 130 by both IL-6 and IL-11 requires two distinct binding epitopes

J Immunol. 1999 Feb 1;162(3):1480-7.

Abstract

The coordination and regulation of immune responses are primarily mediated by cytokines that bind to specific cell surface receptors. Glycoprotein 130 (gp130) belongs to the family of class I cytokine receptors and is the common signal-transducing receptor subunit shared by the so-called IL-6 type cytokines (IL-6, IL-11, ciliary neurotrophic factor, leukemia inhibitory factor, oncostatin M, and cardiotrophin-1). The inflammatory cytokines IL-6 and IL-11 induce gp130 homodimerization after binding to their specific alpha receptors, which leads to the activation of the Janus kinase/STAT signal transduction pathway. A molecular model of IL-6/IL-6R/gp130, which is based on the structure of the growth hormone/growth hormone receptor complex, allowed the selection of several amino acids located in the cytokine-binding module of gp130 for mutagenesis. The mutants were analyzed with regard to IL-6- or IL-11-induced STAT activation and ligand binding. It was found that Y190 and F191 are essential for the interaction of gp130 with IL-6 as well as IL-11, suggesting a common mode of recognition of helical cytokines by class I cytokine receptors. Furthermore, the requirement of the gp130 N-terminal Ig-like domain for ligand binding and signal transduction was demonstrated by the use of deletion mutants. Thus, besides the observed analogy to the growth hormone/growth hormone receptor complex, there is a substantial difference in the mechanism of receptor engagement by cytokines that signal via gp130.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antigens, CD / chemistry*
  • Antigens, CD / genetics
  • Antigens, CD / metabolism*
  • Binding Sites
  • COS Cells
  • Cytokine Receptor gp130
  • Epitopes / chemistry
  • Epitopes / genetics
  • Humans
  • Interleukin-11 / chemistry
  • Interleukin-11 / metabolism
  • Interleukin-11 / pharmacology*
  • Interleukin-11 Receptor alpha Subunit
  • Interleukin-6 / chemistry
  • Interleukin-6 / metabolism
  • Interleukin-6 / pharmacology*
  • Macromolecular Substances
  • Membrane Glycoproteins / chemistry*
  • Membrane Glycoproteins / genetics
  • Membrane Glycoproteins / metabolism*
  • Models, Molecular
  • Mutagenesis, Site-Directed
  • Protein Conformation
  • Receptors, Interleukin / chemistry
  • Receptors, Interleukin / metabolism
  • Receptors, Interleukin-11
  • Receptors, Interleukin-6 / chemistry
  • Receptors, Interleukin-6 / metabolism
  • Signal Transduction

Substances

  • Antigens, CD
  • Epitopes
  • IL11RA protein, human
  • IL6ST protein, human
  • Interleukin-11
  • Interleukin-11 Receptor alpha Subunit
  • Interleukin-6
  • Macromolecular Substances
  • Membrane Glycoproteins
  • Receptors, Interleukin
  • Receptors, Interleukin-11
  • Receptors, Interleukin-6
  • Cytokine Receptor gp130