Ellman JA - Search Results

1

Potent, low-molecular-weight non-peptide inhibitors of malarial aspartyl protease plasmepsin II.

Haque TS, Skillman AG, Lee CE, Habashita H, Gluzman IY, Ewing TJ, Goldberg DE, Kuntz ID, Ellman JA. Haque TS, et al. Among authors: ellman ja. J Med Chem. 1999 Apr 22;42(8):1428-40. doi: 10.1021/jm980641t. J Med Chem. 1999. PMID: 10212129

2

Expedient method for the solid-phase synthesis of aspartic acid protease inhibitors directed toward the generation of libraries.

Kick EK, Ellman JA. Kick EK, et al. Among authors: ellman ja. J Med Chem. 1995 Apr 28;38(9):1427-30. doi: 10.1021/jm00009a002. J Med Chem. 1995. PMID: 7739000 No abstract available.

3

Structure-based design and combinatorial chemistry yield low nanomolar inhibitors of cathepsin D.

Kick EK, Roe DC, Skillman AG, Liu G, Ewing TJ, Sun Y, Kuntz ID, Ellman JA. Kick EK, et al. Among authors: ellman ja. Chem Biol. 1997 Apr;4(4):297-307. doi: 10.1016/s1074-5521(97)90073-9. Chem Biol. 1997. PMID: 9195867

4

Novel inhibitors of alpha 4 beta 1 integrin receptor interactions through library synthesis and screening.

Souers AJ, Virgilio AA, Schürer SS, Ellman JA, Kogan TP, West HE, Ankener W, Vanderslice P. Souers AJ, et al. Among authors: ellman ja. Bioorg Med Chem Lett. 1998 Sep 8;8(17):2297-302. doi: 10.1016/s0960-894x(98)00416-8. Bioorg Med Chem Lett. 1998. PMID: 9873531

5

Combinatorial target-guided ligand assembly: identification of potent subtype-selective c-Src inhibitors.

Maly DJ, Choong IC, Ellman JA. Maly DJ, et al. Among authors: ellman ja. Proc Natl Acad Sci U S A. 2000 Mar 14;97(6):2419-24. doi: 10.1073/pnas.97.6.2419. Proc Natl Acad Sci U S A. 2000. PMID: 10716979 Free PMC article.

6

Novel cathepsin D inhibitors block the formation of hyperphosphorylated tau fragments in hippocampus.

Bi X, Haque TS, Zhou J, Skillman AG, Lin B, Lee CE, Kuntz ID, Ellman JA, Lynch G. Bi X, et al. Among authors: ellman ja. J Neurochem. 2000 Apr;74(4):1469-77. doi: 10.1046/j.1471-4159.2000.0741469.x. J Neurochem. 2000. PMID: 10737603 Free article.

7

Parallel synthesis of prostaglandin E1 analogues.

Dragoli DR, Thompson LA, O'Brien J, Ellman JA. Dragoli DR, et al. Among authors: ellman ja. J Comb Chem. 1999 Nov-Dec;1(6):534-9. doi: 10.1021/cc990033e. J Comb Chem. 1999. PMID: 10748730

8

Optimization of a somatostatin mimetic via constrained amino acid and backbone incorporation.

Souers AJ, Rosenquist A, Jarvie EM, Ladlow M, Feniuk W, Ellman JA. Souers AJ, et al. Among authors: ellman ja. Bioorg Med Chem Lett. 2000 Dec 18;10(24):2731-3. doi: 10.1016/s0960-894x(00)00552-7. Bioorg Med Chem Lett. 2000. PMID: 11133079

9

Definition of the extended substrate specificity determinants for beta-tryptases I and II.

Harris JL, Niles A, Burdick K, Maffitt M, Backes BJ, Ellman JA, Kuntz I, Haak-Frendscho M, Craik CS. Harris JL, et al. Among authors: ellman ja. J Biol Chem. 2001 Sep 14;276(37):34941-7. doi: 10.1074/jbc.M102997200. Epub 2001 Jul 3. J Biol Chem. 2001. PMID: 11438529 Free article.

10

Identification of potent and selective mechanism-based inhibitors of the cysteine protease cruzain using solid-phase parallel synthesis.

Huang L, Lee A, Ellman JA. Huang L, et al. Among authors: ellman ja. J Med Chem. 2002 Jan 31;45(3):676-84. doi: 10.1021/jm010333m. J Med Chem. 2002. PMID: 11806719

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