Wheeldon A - Search Results

1

The substance P antagonist L-760,735 inhibits stress-induced NK(1) receptor internalisation in the basolateral amygdala.

Smith DW, Hewson L, Fuller P, Williams AR, Wheeldon A, Rupniak NM. Smith DW, et al. Among authors: wheeldon a. Brain Res. 1999 Nov 27;848(1-2):90-5. doi: 10.1016/s0006-8993(99)01976-9. Brain Res. 1999. PMID: 10612700

2

Pharmacological blockade or genetic deletion of substance P (NK(1)) receptors attenuates neonatal vocalisation in guinea-pigs and mice.

Rupniak NM, Carlson EC, Harrison T, Oates B, Seward E, Owen S, de Felipe C, Hunt S, Wheeldon A. Rupniak NM, et al. Among authors: wheeldon a. Neuropharmacology. 2000 Jun 8;39(8):1413-21. doi: 10.1016/s0028-3908(00)00052-6. Neuropharmacology. 2000. PMID: 10818257

3

Comparison of the phenotype of NK1R-/- mice with pharmacological blockade of the substance P (NK1 ) receptor in assays for antidepressant and anxiolytic drugs.

Rupniak NM, Carlson EJ, Webb JK, Harrison T, Porsolt RD, Roux S, de Felipe C, Hunt SP, Oates B, Wheeldon A. Rupniak NM, et al. Among authors: wheeldon a. Behav Pharmacol. 2001 Nov;12(6-7):497-508. doi: 10.1097/00008877-200111000-00011. Behav Pharmacol. 2001. PMID: 11742144

4

Chronic substance P (NK1) receptor antagonist and conventional antidepressant treatment increases burst firing of monoamine neurones in the locus coeruleus.

Maubach KA, Martin K, Chicchi G, Harrison T, Wheeldon A, Swain CJ, Cumberbatch MJ, Rupniak NM, Seabrook GR. Maubach KA, et al. Among authors: wheeldon a. Neuroscience. 2002;109(3):609-17. doi: 10.1016/s0306-4522(01)00467-5. Neuroscience. 2002. PMID: 11823070

5

Fused bicyclic pyrrolizinones as new scaffolds for human NK1 antagonists.

Morriello GJ, Devita RJ, Mills SG, Young JR, Lin P, Doss G, Chicchi GG, Demartino J, Kurtz MM, Tsao KL, Carlson E, Townson K, Wheeldon A, Boyce S, Collinson N, Rupniak N, Moore S. Morriello GJ, et al. Among authors: wheeldon a. Bioorg Med Chem. 2008 Mar 1;16(5):2156-70. doi: 10.1016/j.bmc.2007.11.081. Epub 2007 Dec 5. Bioorg Med Chem. 2008. PMID: 18248994

6

Fused tricyclic pyrrolizinones that exhibit pseudo-irreversible blockade of the NK1 receptor.

Morriello GJ, Chicchi G, Johnson T, Mills SG, Demartino J, Kurtz M, Tsao KL, Zheng S, Tong X, Carlson E, Townson K, Wheeldon A, Boyce S, Collinson N, Rupniak N, Devita RJ. Morriello GJ, et al. Among authors: wheeldon a. Bioorg Med Chem Lett. 2010 Oct 1;20(19):5925-32. doi: 10.1016/j.bmcl.2010.07.058. Epub 2010 Jul 19. Bioorg Med Chem Lett. 2010. PMID: 20729082

7

Substituted fused bicyclic pyrrolizinones as potent, orally bioavailable hNK1 antagonists.

Morriello GJ, Mills SG, Johnson T, Reibarkh M, Chicchi G, DeMartino J, Kurtz M, Davies P, Tsao KL, Zheng S, Tong X, Carlson E, Townson K, Tattersall FD, Wheeldon A, Boyce S, Collinson N, Rupniak N, Moore S, DeVita RJ. Morriello GJ, et al. Among authors: wheeldon a. Bioorg Med Chem Lett. 2010 Mar 15;20(6):2007-12. doi: 10.1016/j.bmcl.2010.01.065. Epub 2010 Jan 20. Bioorg Med Chem Lett. 2010. PMID: 20153964

8

1-Phenyl-8-azabicyclo[3.2.1]octane ethers: a novel series of neurokinin (NK1) antagonists.

Huscroft IT, Carlson EJ, Chicchi GG, Kurtz MM, London C, Raubo P, Wheeldon A, Kulagowski JJ. Huscroft IT, et al. Among authors: wheeldon a. Bioorg Med Chem Lett. 2006 Apr 1;16(7):2008-12. doi: 10.1016/j.bmcl.2005.12.069. Epub 2006 Jan 18. Bioorg Med Chem Lett. 2006. PMID: 16413782

9

Inhibition of acute nociceptive responses in rat spinal cord by a bradykinin B1 receptor antagonist.

Conley RK, Wheeldon A, Webb JK, DiPardo RM, Homnick CF, Bock MG, Chen TB, Chang RS, Pettibone DJ, Boyce S. Conley RK, et al. Among authors: wheeldon a. Eur J Pharmacol. 2005 Dec 19;527(1-3):44-51. doi: 10.1016/j.ejphar.2005.06.057. Epub 2005 Nov 28. Eur J Pharmacol. 2005. PMID: 16310181

10

Tetrahydroindolizinone NK1 antagonists.

Bao J, Lu H, Morriello GJ, Carlson EJ, Wheeldon A, Chicchi GG, Kurtz MM, Tsao KL, Zheng S, Tong X, Mills SG, DeVita RJ. Bao J, et al. Among authors: wheeldon a. Bioorg Med Chem Lett. 2010 Apr 1;20(7):2354-8. doi: 10.1016/j.bmcl.2010.01.120. Epub 2010 Feb 1. Bioorg Med Chem Lett. 2010. PMID: 20188553

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