Cheng K - Search Results

1

A potent, nonpeptidyl 1H-quinolone antagonist for the gonadotropin-releasing hormone receptor.

DeVita RJ, Walsh TF, Young JR, Jiang J, Ujjainwalla F, Toupence RB, Parikh M, Huang SX, Fair JA, Goulet MT, Wyvratt MJ, Lo JL, Ren N, Yudkovitz JB, Yang YT, Cheng K, Cui J, Mount G, Rohrer SP, Schaeffer JM, Rhodes L, Drisko JE, McGowan E, MacIntyre DE, Vincent S, Carlin JR, Cameron J, Smith RG. DeVita RJ, et al. Among authors: cheng k. J Med Chem. 2001 Mar 15;44(6):917-22. doi: 10.1021/jm000275p. J Med Chem. 2001. PMID: 11300873

2

A potent, orally bioavailable benzazepinone growth hormone secretagogue.

DeVita RJ, Bochis R, Frontier AJ, Kotliar A, Fisher MH, Schoen WR, Wyvratt MJ, Cheng K, Chan WW, Butler B, Jacks TM, Hickey GJ, Schleim KD, Leung K, Chen Z, Chiu SL, Feeney WP, Cunningham PK, Smith RG. DeVita RJ, et al. Among authors: cheng k. J Med Chem. 1998 May 7;41(10):1716-28. doi: 10.1021/jm970816j. J Med Chem. 1998. PMID: 9572898

3

Spiro[1H-indene-1,4'-piperidine] derivatives as potent and selective non-peptide human somatostatin receptor subtype 2 (sst2) agonists.

Yang L, Guo L, Pasternak A, Mosley R, Rohrer S, Birzin E, Foor F, Cheng K, Schaeffer J, Patchett AA. Yang L, et al. Among authors: cheng k. J Med Chem. 1998 Jun 18;41(13):2175-9. doi: 10.1021/jm980194h. J Med Chem. 1998. PMID: 9632348 No abstract available.

4

Identification and initial structure-activity relationships of a novel non-peptide quinolone GnRH receptor antagonist.

DeVita RJ, Hollings DD, Goulet MT, Wyvratt MJ, Fisher MH, Lo JL, Yang YT, Cheng K, Smith RG. DeVita RJ, et al. Among authors: cheng k. Bioorg Med Chem Lett. 1999 Sep 6;9(17):2615-20. doi: 10.1016/s0960-894x(99)00446-1. Bioorg Med Chem Lett. 1999. PMID: 10498220

5

Investigation of the 4-O-alkylamine substituent of non-peptide quinolone GnRH receptor antagonists.

DeVita RJ, Goulet MT, Wyvratt MJ, Fisher MH, Lo JL, Yang YT, Cheng K, Smith RG. DeVita RJ, et al. Among authors: cheng k. Bioorg Med Chem Lett. 1999 Sep 6;9(17):2621-4. doi: 10.1016/s0960-894x(99)00447-3. Bioorg Med Chem Lett. 1999. PMID: 10498221

6

Acyclic structural variants of growth hormone secretagogue L-692,429.

Lin P, Pisano JM, Schoen WR, Cheng K, Chan WW, Butler BS, Smith RG, Fisher MH, Wyvratt MJ. Lin P, et al. Among authors: cheng k. Bioorg Med Chem Lett. 1999 Nov 15;9(22):3237-42. doi: 10.1016/s0960-894x(99)00568-5. Bioorg Med Chem Lett. 1999. PMID: 10576695

7

Potent antagonists of gonadotropin releasing hormone receptors derived from quinolone-6-carboxamides.

Walsh TF, Toupence RB, Young JR, Huang SX, Ujjainwalla F, DeVita RJ, Goulet MT, Wyvratt MJ Jr, Fisher MH, Lo JL, Ren N, Yudkovitz JB, Yang YT, Cheng K, Smith RG. Walsh TF, et al. Among authors: cheng k. Bioorg Med Chem Lett. 2000 Mar 6;10(5):443-7. doi: 10.1016/s0960-894x(00)00024-x. Bioorg Med Chem Lett. 2000. PMID: 10743944

8

Identification of Phe313 of the gonadotropin-releasing hormone (GnRH) receptor as a site critical for the binding of nonpeptide GnRH antagonists.

Cui J, Smith RG, Mount GR, Lo JL, Yu J, Walsh TF, Singh SB, DeVita RJ, Goulet MT, Schaeffer JM, Cheng K. Cui J, et al. Among authors: cheng k. Mol Endocrinol. 2000 May;14(5):671-81. doi: 10.1210/mend.14.5.0464. Mol Endocrinol. 2000. PMID: 10809231

9

Quinolones as gonadotropin releasing hormone (GnRH) antagonists: simultaneous optimization of the C(3)-aryl and C(6)-substituents.

Young JR, Huang SX, Chen I, Walsh TF, DeVita RJ, Wyvratt MJ Jr, Goulet MT, Ren N, Lo J, Yang YT, Yudkovitz JB, Cheng K, Smith RG. Young JR, et al. Among authors: cheng k. Bioorg Med Chem Lett. 2000 Aug 7;10(15):1723-7. doi: 10.1016/s0960-894x(00)00318-8. Bioorg Med Chem Lett. 2000. PMID: 10937733

10

Nipecotic and iso-nipecotic amides as potent and selective somatostatin subtype-2 receptor agonists.

Zhou C, Guo L, Morriello G, Pasternak A, Pan Y, Rohrer SP, Birzin ET, Huskey SE, Jacks T, Schleim KD, Cheng K, Schaeffer JM, Patchett AA, Yang L. Zhou C, et al. Among authors: cheng k. Bioorg Med Chem Lett. 2001 Feb 12;11(3):415-7. doi: 10.1016/s0960-894x(00)00687-9. Bioorg Med Chem Lett. 2001. PMID: 11212124

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