De Clercq E - Search Results

1

Design, synthesis and enzymatic activity of highly selective human mitochondrial thymidine kinase inhibitors.

Manfredini S, Baraldi PG, Durini E, Porcu L, Angusti A, Vertuani S, Solaroli N, De Clercq E, Karlsson A, Balzarini J. Manfredini S, et al. Among authors: de clercq e. Bioorg Med Chem Lett. 2001 May 21;11(10):1329-32. doi: 10.1016/s0960-894x(01)00207-4. Bioorg Med Chem Lett. 2001. PMID: 11392548

2

Geiparvarin analogues. 2. Synthesis and cytostatic activity of 5-(4-arylbutadienyl)-3(2H)-furanones and of N-substituted 3-(4-oxo-2-furanyl)-2-buten-2-yl carbamates.

Simoni D, Manfredini S, Tabrizi MA, Bazzanini R, Baraldi PG, Balzarini J, De Clercq E. Simoni D, et al. Among authors: de clercq e. J Med Chem. 1991 Nov;34(11):3172-6. doi: 10.1021/jm00115a004. J Med Chem. 1991. PMID: 1956034

3

Synthesis and cytostatic activity of geiparvarin analogues.

Baraldi PG, Guarneri M, Manfredini S, Simoni D, Balzarini J, De Clercq E. Baraldi PG, et al. Among authors: de clercq e. J Med Chem. 1989 Feb;32(2):284-8. doi: 10.1021/jm00122a002. J Med Chem. 1989. PMID: 2913291

4

Synthesis and cytotoxic activity of 6-vinyl- and 6-ethynyluridine and 8-vinyl-and 8-ethynyladenosine.

Manfredini S, Baraldi PG, Bazzanini R, Marangoni M, Simoni D, Balzarini J, De Clercq E. Manfredini S, et al. Among authors: de clercq e. J Med Chem. 1995 Jan 6;38(1):199-203. doi: 10.1021/jm00001a025. J Med Chem. 1995. PMID: 7837231

5

Geiparvarin analogues. 4. Synthesis and cytostatic activity of geiparvarin analogues bearing a carbamate moiety or a furocoumarin fragment on the alkenyl side chain.

Manfredini S, Baraldi PG, Bazzanini R, Guarneri M, Simoni D, Balzarini J, De Clercq E. Manfredini S, et al. Among authors: de clercq e. J Med Chem. 1994 Jul 22;37(15):2401-5. doi: 10.1021/jm00041a019. J Med Chem. 1994. PMID: 8057288

6

5'-Phosphoramidates and 5'-diphosphates of 2'-O-allyl-beta-D-arabinofuranosyluracil, -cytosine, and -adenine: inhibition of ribonucleotide reductase.

Manfredini S, Baraldi PG, Durini E, Vertuani S, Balzarini J, De Clercq E, Karlsson A, Buzzoni V, Thelander L. Manfredini S, et al. Among authors: de clercq e. J Med Chem. 1999 Aug 26;42(17):3243-50. doi: 10.1021/jm9807095. J Med Chem. 1999. PMID: 10464011

7

Geiparvarin analogues. 3. Synthesis and cytostatic activity of 3(2H)-furanone and 4,5-dihydro-3(2H)-furanone congeners of geiparvarin, containing a geraniol-like fragment in the side chain.

Baraldi PG, Manfredini S, Simoni D, Tabrizi MA, Balzarini J, De Clercq E. Baraldi PG, et al. Among authors: de clercq e. J Med Chem. 1992 May 15;35(10):1877-82. doi: 10.1021/jm00088a025. J Med Chem. 1992. PMID: 1588564

8

Retinoic acid conjugates as potential antitumor agents: synthesis and biological activity of conjugates with Ara-A, Ara-C, 3(2H)-furanone, and aniline mustard moieties.

Manfredini S, Simoni D, Ferroni R, Bazzanini R, Vertuani S, Hatse S, Balzarini J, De Clercq E. Manfredini S, et al. Among authors: de clercq e. J Med Chem. 1997 Nov 7;40(23):3851-7. doi: 10.1021/jm9602322. J Med Chem. 1997. PMID: 9371251

9

Synthesis, cytostatic activity and inhibition of ribonucleotide reductase by 5'-phosphoramidates and 5'-diphosphates, of 2'-O-allyl-arabinofuranosyl nucleosides.

Manfredini S, Baraldi PG, Durini E, Balzarini J, De Clercq E, Karlsson A, Buzzoni V, Thelander L. Manfredini S, et al. Among authors: de clercq e. Nucleosides Nucleotides. 1999 Apr-May;18(4-5):1007-8. doi: 10.1080/15257779908041631. Nucleosides Nucleotides. 1999. PMID: 10432732

10

Design, synthesis, and enzymatic evaluation of multisubstrate analogue inhibitors of Escherichia coli thymidine phosphorylase.

Esteban-Gamboa A, Balzarini J, Esnouf R, De Clercq E, Camarasa MJ, Pérez-Pérez MJ. Esteban-Gamboa A, et al. Among authors: de clercq e. J Med Chem. 2000 Mar 9;43(5):971-83. doi: 10.1021/jm9911377. J Med Chem. 2000. PMID: 10715161

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