Becker B - Search Results

1

Original 2-alkylamino-6-halogenoquinazolin-4(3H)-ones and K(ATP) channel activity.

Somers F, Ouedraogo R, Antoine MH, de Tullio P, Becker B, Fontaine J, Damas J, Dupont L, Rigo B, Delarge J, Lebrun P, Pirotte B. Somers F, et al. Among authors: becker b. J Med Chem. 2001 Aug 2;44(16):2575-85. doi: 10.1021/jm0004648. J Med Chem. 2001. PMID: 11472211

2

2-alkyl-3-Alkylamino-2H-Benzo- and pyridothiadiazine 1,1-dioxides: from K+ATP channel openers to Ca++ channel blockers?

Ouedraogo R, Becker B, Boverie S, Somers F, Antoine MH, Pirotte B, Lebrun P, de Tullio P. Ouedraogo R, et al. Among authors: becker b. Biol Chem. 2002 Nov;383(11):1759-68. doi: 10.1515/BC.2002.197. Biol Chem. 2002. PMID: 12530541

3

Toward tissue-selective pancreatic B-cells KATP channel openers belonging to 3-alkylamino-7-halo-4H-1,2,4-benzothiadiazine 1,1-dioxides.

de Tullio P, Becker B, Boverie S, Dabrowski M, Wahl P, Antoine MH, Somers F, Sebille S, Ouedraogo R, Hansen JB, Lebrun P, Pirotte B. de Tullio P, et al. Among authors: becker b. J Med Chem. 2003 Jul 17;46(15):3342-53. doi: 10.1021/jm021117w. J Med Chem. 2003. PMID: 12852765

4

4,6-Disubstituted 2,2-dimethylchromans structurally related to the K(ATP) channel opener cromakalim: design, synthesis, and effect on insulin release and vascular tone.

Sebille S, de Tullio P, Becker B, Antoine MH, Boverie S, Pirotte B, Lebrun P. Sebille S, et al. Among authors: becker b. J Med Chem. 2005 Jan 27;48(2):614-21. doi: 10.1021/jm040789e. J Med Chem. 2005. PMID: 15658874

5

Effect on K(ATP) channel activation properties and tissue selectivity of the nature of the substituent in the 7- and the 3-position of 4H-1,2,4-benzothiadiazine 1,1-dioxides.

Boverie S, Antoine MH, Somers F, Becker B, Sebille S, Ouedraogo R, Counerotte S, Pirotte B, Lebrun P, de Tullio P. Boverie S, et al. Among authors: becker b. J Med Chem. 2005 May 19;48(10):3492-503. doi: 10.1021/jm0311339. J Med Chem. 2005. PMID: 15887958

6

3-Alkylamino-4H-1,2,4-benzothiadiazine 1,1-dioxides as ATP-sensitive potassium channel openers: effect of 6,7-disubstitution on potency and tissue selectivity.

de Tullio P, Boverie S, Becker B, Antoine MH, Nguyen QA, Francotte P, Counerotte S, Sebille S, Pirotte B, Lebrun P. de Tullio P, et al. Among authors: becker b. J Med Chem. 2005 Jul 28;48(15):4990-5000. doi: 10.1021/jm0580050. J Med Chem. 2005. PMID: 16033278

7

New R/S-3,4-dihydro-2,2-dimethyl-6-halo-4-(phenylaminothiocarbonylamino)-2H-1-benzopyrans structurally related to (+/-)-cromakalim as tissue-selective pancreatic beta-cell K(ATP) channel openers.

Sebille S, de Tullio P, Florence X, Becker B, Antoine MH, Michaux C, Wouters J, Pirotte B, Lebrun P. Sebille S, et al. Among authors: becker b. Bioorg Med Chem. 2008 May 15;16(10):5704-19. doi: 10.1016/j.bmc.2008.03.065. Epub 2008 Mar 30. Bioorg Med Chem. 2008. PMID: 18406154

8

Effect on insulin release of compounds structurally related to the potassium-channel opener 7-chloro-3-isopropylamino-4H-1,2,4-benzothiadiazine 1,1-dioxide (BPDZ 73): introduction of heteroatoms on the 3-alkylamino side chain of the benzothiadiazine 1,1-dioxide ring.

Boverie S, Antoine MH, de Tullio P, Somers F, Becker B, Sebille S, Lebrun P, Pirotte B. Boverie S, et al. Among authors: becker b. J Pharm Pharmacol. 2001 Jul;53(7):973-80. doi: 10.1211/0022357011776216. J Pharm Pharmacol. 2001. PMID: 11480549

9

Synthesis and characterization of a quinolinonic compound activating ATP-sensitive K(+) channels in endocrine and smooth muscle tissues.

Becker B, Antoine MH, Nguyen QA, Rigo B, Cosgrove KE, Barnes PD, Dunne MJ, Pirotte B, Lebrun P. Becker B, et al. Br J Pharmacol. 2001 Sep;134(2):375-85. doi: 10.1038/sj.bjp.0704266. Br J Pharmacol. 2001. PMID: 11564656 Free PMC article.

10

KATP channel openers: tissue selectivity of original 3-alkylaminopyrido- and 3-alkylaminobenzothiadiazine 1,1-dioxides.

Lebrun P, Becker B, Morel N, Ghisdal P, Antoine MH, de Tullio P, Pirotte B. Lebrun P, et al. Among authors: becker b. Biochem Pharmacol. 2008 Jan 15;75(2):468-75. doi: 10.1016/j.bcp.2007.08.032. Epub 2007 Sep 1. Biochem Pharmacol. 2008. PMID: 17920043

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