Sausville EA - Search Results

1

Aryl hydrocarbon receptor mediates sensitivity of MCF-7 breast cancer cells to antitumor agent 2-(4-amino-3-methylphenyl) benzothiazole.

Loaiza-Pérez AI, Trapani V, Hose C, Singh SS, Trepel JB, Stevens MF, Bradshaw TD, Sausville EA. Loaiza-Pérez AI, et al. Among authors: sausville ea. Mol Pharmacol. 2002 Jan;61(1):13-9. doi: 10.1124/mol.61.1.13. Mol Pharmacol. 2002. PMID: 11752201

2

Preclinical evaluation of amino acid prodrugs of novel antitumor 2-(4-amino-3-methylphenyl)benzothiazoles.

Bradshaw TD, Bibby MC, Double JA, Fichtner I, Cooper PA, Alley MC, Donohue S, Stinson SF, Tomaszewjski JE, Sausville EA, Stevens MF. Bradshaw TD, et al. Among authors: sausville ea. Mol Cancer Ther. 2002 Feb;1(4):239-46. Mol Cancer Ther. 2002. PMID: 12467219

3

Genotoxic profiling of MCF-7 breast cancer cell line elucidates gene expression modifications underlying toxicity of the anticancer drug 2-(4-amino-3-methylphenyl)-5-fluorobenzothiazole.

Monks A, Harris E, Hose C, Connelly J, Sausville EA. Monks A, et al. Among authors: sausville ea. Mol Pharmacol. 2003 Mar;63(3):766-72. doi: 10.1124/mol.63.3.766. Mol Pharmacol. 2003. PMID: 12606787

4

Induction of CYP1A1 in tumor cells by the antitumor agent 2-[4-amino-3-methylphenyl]-5-fluoro-benzothiazole: a potential surrogate marker for patient sensitivity.

Hose CD, Hollingshead M, Sausville EA, Monks A. Hose CD, et al. Among authors: sausville ea. Mol Cancer Ther. 2003 Dec;2(12):1265-72. Mol Cancer Ther. 2003. PMID: 14707267

5

Aryl hydrocarbon receptor activation of an antitumor aminoflavone: basis of selective toxicity for MCF-7 breast tumor cells.

Loaiza-Pérez AI, Kenney S, Boswell J, Hollingshead M, Alley MC, Hose C, Ciolino HP, Yeh GC, Trepel JB, Vistica DT, Sausville EA. Loaiza-Pérez AI, et al. Among authors: sausville ea. Mol Cancer Ther. 2004 Jun;3(6):715-25. Mol Cancer Ther. 2004. PMID: 15210858

6

Fluorinated 2-(4-amino-3-methylphenyl)benzothiazoles induce CYP1A1 expression, become metabolized, and bind to macromolecules in sensitive human cancer cells.

Brantley E, Trapani V, Alley MC, Hose CD, Bradshaw TD, Stevens MF, Sausville EA, Stinson SF. Brantley E, et al. Among authors: sausville ea. Drug Metab Dispos. 2004 Dec;32(12):1392-401. doi: 10.1124/dmd.104.001057. Epub 2004 Sep 8. Drug Metab Dispos. 2004. PMID: 15355884

7

The antitumor drug candidate 2-(4-amino-3-methylphenyl)-5-fluorobenzothiazole induces NF-kappaB activity in drug-sensitive MCF-7 cells.

Brantley E, Patel V, Stinson SF, Trapani V, Hose CD, Ciolino HP, Yeh GC, Gutkind JS, Sausville EA, Loaiza-Pérez AI. Brantley E, et al. Among authors: sausville ea. Anticancer Drugs. 2005 Feb;16(2):137-43. doi: 10.1097/00001813-200502000-00004. Anticancer Drugs. 2005. PMID: 15655410

8

Role of Cyp1A1 in modulation of antitumor properties of the novel agent 2-(4-amino-3-methylphenyl)benzothiazole (DF 203, NSC 674495) in human breast cancer cells.

Chua MS, Kashiyama E, Bradshaw TD, Stinson SF, Brantley E, Sausville EA, Stevens MF. Chua MS, et al. Among authors: sausville ea. Cancer Res. 2000 Sep 15;60(18):5196-203. Cancer Res. 2000. PMID: 11016648

9

Transcriptional regulation of the transforming growth factor beta type II receptor gene by histone acetyltransferase and deacetylase is mediated by NF-Y in human breast cancer cells.

Park SH, Lee SR, Kim BC, Cho EA, Patel SP, Kang HB, Sausville EA, Nakanishi O, Trepel JB, Lee BI, Kim SJ. Park SH, et al. Among authors: sausville ea. J Biol Chem. 2002 Feb 15;277(7):5168-74. doi: 10.1074/jbc.M106451200. Epub 2001 Dec 13. J Biol Chem. 2002. PMID: 11744689 Free article.

10

Perifosine, a novel alkylphospholipid, inhibits protein kinase B activation.

Kondapaka SB, Singh SS, Dasmahapatra GP, Sausville EA, Roy KK. Kondapaka SB, et al. Among authors: sausville ea. Mol Cancer Ther. 2003 Nov;2(11):1093-103. Mol Cancer Ther. 2003. PMID: 14617782

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