Brasili L - Search Results

1

Alpha2-adrenoreceptors profile modulation and high antinociceptive activity of (S)-(-)-2-[1-(biphenyl-2-yloxy)ethyl]-4,5-dihydro-1H-imidazole.

Gentili F, Bousquet P, Brasili L, Caretto M, Carrieri A, Dontenwill M, Giannella M, Marucci G, Perfumi M, Piergentili A, Quaglia W, Rascente C, Pigini M. Gentili F, et al. Among authors: brasili l. J Med Chem. 2002 Jan 3;45(1):32-40. doi: 10.1021/jm0110082. J Med Chem. 2002. PMID: 11754577

2

Imidazoline binding sites (IBS) profile modulation: key role of the bridge in determining I1-IBS or I2-IBS selectivity within a series of 2-phenoxymethylimidazoline analogues.

Gentili F, Bousquet P, Brasili L, Dontenwill M, Feldman J, Ghelfi F, Giannella M, Piergentili A, Quaglia W, Pigini M. Gentili F, et al. Among authors: brasili l. J Med Chem. 2003 May 22;46(11):2169-76. doi: 10.1021/jm021113r. J Med Chem. 2003. PMID: 12747788

3

Structure-activity relationships in 1,4-benzodioxan-related compounds. Investigation on the role of the dehydrodioxane ring on alpha 1-adrenoreceptor blocking activity.

Pigini M, Brasili L, Giannella M, Giardinà D, Gulini U, Quaglia W, Melchiorre C. Pigini M, et al. Among authors: brasili l. J Med Chem. 1988 Dec;31(12):2300-4. doi: 10.1021/jm00120a009. J Med Chem. 1988. PMID: 2903932

4

Separation of alpha-adrenergic and imidazoline/guanidinium receptive sites (IGRS) activity in a series of imidazoline analogues of cirazoline.

Brasili L, Pigini M, Marucci G, Quaglia W, Malmusi L, Lanier SM, Lanier B. Brasili L, et al. Bioorg Med Chem. 1995 Nov;3(11):1503-9. doi: 10.1016/0968-0896(95)00132-z. Bioorg Med Chem. 1995. PMID: 8634830

5

Synthesis and structure-activity relationship studies in a series of 2-substituted 1,3-dioxolanes modified at the cationic head.

Angeli P, Brasili L, Cingolani ML, Marucci G, Piergentili A, Pigini M, Quaglia W. Angeli P, et al. Among authors: brasili l. Bioorg Med Chem. 1997 Apr;5(4):731-7. doi: 10.1016/s0968-0896(97)00017-5. Bioorg Med Chem. 1997. PMID: 9158872

6

Imidazoline receptors: qualitative structure-activity relationships and discovery of tracizoline and benazoline. Two ligands with high affinity and unprecedented selectivity.

Pigini M, Bousquet P, Carotti A, Dontenwill M, Giannella M, Moriconi R, Piergentili A, Quaglia W, Tayebati SK, Brasili L. Pigini M, et al. Among authors: brasili l. Bioorg Med Chem. 1997 May;5(5):833-41. doi: 10.1016/s0968-0896(97)00009-6. Bioorg Med Chem. 1997. PMID: 9208095

7

2-D and 3-D modeling of imidazoline receptor ligands: insights into pharmacophore.

Carrieri A, Brasili L, Leonetti F, Pigini M, Giannella M, Bousquet P, Carotti A. Carrieri A, et al. Among authors: brasili l. Bioorg Med Chem. 1997 May;5(5):843-56. doi: 10.1016/s0968-0896(97)00023-0. Bioorg Med Chem. 1997. PMID: 9208096

8

1'-Benzyl-3,4-dihydrospiro[2H-1- benzothiopyran-2,4'-piperidine] (spipethiane), a potent and highly selective sigma1 ligand.

Quaglia W, Giannella M, Piergentili A, Pigini M, Brasili L, Di Toro R, Rossetti L, Spampinato S, Melchiorre C. Quaglia W, et al. Among authors: brasili l. J Med Chem. 1998 May 7;41(10):1557-60. doi: 10.1021/jm970740r. J Med Chem. 1998. PMID: 9572880 No abstract available.

9

Ligand binding to I2 imidazoline receptor: the role of lipophilicity in quantitative structure-activity relationship models.

Pigini M, Bousquet P, Brasili L, Carrieri A, Cavagna R, Dontenwill M, Gentili F, Giannella M, Leonetti F, Piergentili A, Quaglia W, Carotti A. Pigini M, et al. Among authors: brasili l. Bioorg Med Chem. 1998 Dec;6(12):2245-60. doi: 10.1016/s0968-0896(98)80005-9. Bioorg Med Chem. 1998. PMID: 9925287

10

2-(2-Phenylcyclopropyl)imidazolines: reversed enantioselective interaction at I(1) and I(2) imidazoline receptors.

Quaglia W, Bousquet P, Pigini M, Carotti A, Carrieri A, Dontenwill M, Gentili F, Giannella M, Maranca F, Piergentili A, Brasili L. Quaglia W, et al. Among authors: brasili l. J Med Chem. 1999 Jul 29;42(15):2737-40. doi: 10.1021/jm991049m. J Med Chem. 1999. PMID: 10425083 No abstract available.

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