Thompson JE - Search Results

1

Photochemical preparation of a pyridone containing tetracycle: a Jak protein kinase inhibitor.

Thompson JE, Cubbon RM, Cummings RT, Wicker LS, Frankshun R, Cunningham BR, Cameron PM, Meinke PT, Liverton N, Weng Y, DeMartino JA. Thompson JE, et al. Bioorg Med Chem Lett. 2002 Apr 22;12(8):1219-23. doi: 10.1016/s0960-894x(02)00106-3. Bioorg Med Chem Lett. 2002. PMID: 11934592

2

Hybrid-designed inhibitors of p38 MAP kinase utilizing N-arylpyridazinones.

Colletti SL, Frie JL, Dixon EC, Singh SB, Choi BK, Scapin G, Fitzgerald CE, Kumar S, Nichols EA, O'Keefe SJ, O'Neill EA, Porter G, Samuel K, Schmatz DM, Schwartz CD, Shoop WL, Thompson CM, Thompson JE, Wang R, Woods A, Zaller DM, Doherty JB. Colletti SL, et al. Among authors: thompson je, thompson cm. J Med Chem. 2003 Jan 30;46(3):349-52. doi: 10.1021/jm025585h. J Med Chem. 2003. PMID: 12540232

3

Mechanism of Janus kinase 3-catalyzed phosphorylation of a Janus kinase 1 activation loop peptide.

Wang R, Griffin PR, Small EC, Thompson JE. Wang R, et al. Among authors: thompson je. Arch Biochem Biophys. 2003 Feb 1;410(1):7-15. doi: 10.1016/s0003-9861(02)00637-9. Arch Biochem Biophys. 2003. PMID: 12559972

4

p38 Inhibitors: piperidine- and 4-aminopiperidine-substituted naphthyridinones, quinolinones, and dihydroquinazolinones.

Hunt JA, Kallashi F, Ruzek RD, Sinclair PJ, Ita I, McCormick SX, Pivnichny JV, Hop CE, Kumar S, Wang Z, O'Keefe SJ, O'Neill EA, Porter G, Thompson JE, Woods A, Zaller DM, Doherty JB. Hunt JA, et al. Among authors: thompson je. Bioorg Med Chem Lett. 2003 Feb 10;13(3):467-70. doi: 10.1016/s0960-894x(02)00990-3. Bioorg Med Chem Lett. 2003. PMID: 12565952

5

Time-resolved Forster resonance energy transfer assays for the binding of nucleotide and protein substrates to p38alpha protein kinase.

Zhang WX, Wang R, Wisniewski D, Marcy AI, LoGrasso P, Lisnock JM, Cummings RT, Thompson JE. Zhang WX, et al. Among authors: thompson je. Anal Biochem. 2005 Aug 1;343(1):76-83. doi: 10.1016/j.ab.2005.05.011. Anal Biochem. 2005. PMID: 15979553

6

JAK protein kinase inhibitors.

Thompson JE. Thompson JE. Drug News Perspect. 2005 Jun;18(5):305-10. doi: 10.1358/dnp.2005.18.5.904198. Drug News Perspect. 2005. PMID: 16193102 Free article. Review.

7

p38 MAP kinase inhibitors: metabolically stabilized piperidine-substituted quinolinones and naphthyridinones.

Bao J, Hunt JA, Miao S, Rupprecht KM, Stelmach JE, Liu L, Ruzek RD, Sinclair PJ, Pivnichny JV, Hop CE, Kumar S, Zaller DM, Shoop WL, O'neill EA, O'keefe SJ, Thompson CM, Cubbon RM, Wang R, Zhang WX, Thompson JE, Doherty JB. Bao J, et al. Among authors: thompson je, thompson cm. Bioorg Med Chem Lett. 2006 Jan 1;16(1):64-8. doi: 10.1016/j.bmcl.2005.09.065. Epub 2005 Oct 18. Bioorg Med Chem Lett. 2006. PMID: 16242322

8

p38 MAP kinase inhibitors. Part 3: SAR on 3,4-dihydropyrimido[4,5-d]pyrimidin-2-ones and 3,4-dihydropyrido[4,3-d]pyrimidin-2-ones.

Natarajan SR, Wisnoski DD, Thompson JE, O'Neill EA, O'Keefe SJ. Natarajan SR, et al. Among authors: thompson je. Bioorg Med Chem Lett. 2006 Aug 15;16(16):4400-4. doi: 10.1016/j.bmcl.2006.05.045. Epub 2006 Jun 5. Bioorg Med Chem Lett. 2006. PMID: 16750629

9

p38 MAP kinase inhibitors. Part 6: 2-arylpyridazin-3-ones as templates for inhibitor design.

Natarajan SR, Heller ST, Nam K, Singh SB, Scapin G, Patel S, Thompson JE, Fitzgerald CE, O'Keefe SJ. Natarajan SR, et al. Among authors: thompson je. Bioorg Med Chem Lett. 2006 Nov 15;16(22):5809-13. doi: 10.1016/j.bmcl.2006.08.074. Epub 2006 Aug 30. Bioorg Med Chem Lett. 2006. PMID: 16945533

10

p38 MAP kinase inhibitors. Part 5: discovery of an orally bio-available and highly efficacious compound based on the 7-amino-naphthyridone scaffold.

Natarajan SR, Liu L, Levorse M, Thompson JE, O'Neill EA, O'Keefe SJ, Vora KA, Cvetovich R, Chung JY, Carballo-Jane E, Visco DM. Natarajan SR, et al. Among authors: thompson je. Bioorg Med Chem Lett. 2006 Oct 15;16(20):5468-71. doi: 10.1016/j.bmcl.2006.06.084. Epub 2006 Sep 1. Bioorg Med Chem Lett. 2006. PMID: 16945534

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