Walters DE - Search Results

1

Novel cyclourethane-derived HIV protease inhibitors: a ring-closing olefin metathesis based strategy.

Ghosh AK, Swanson LM, Liu C, Hussain KA, Cho H, Walters DE, Holland L, Buthod J. Ghosh AK, et al. Among authors: walters de. Bioorg Med Chem Lett. 2002 Aug 5;12(15):1993-6. doi: 10.1016/s0960-894x(02)00300-1. Bioorg Med Chem Lett. 2002. PMID: 12113826

2

Structure-based design: synthesis and biological evaluation of a series of novel cycloamide-derived HIV-1 protease inhibitors.

Ghosh AK, Swanson LM, Cho H, Leshchenko S, Hussain KA, Kay S, Walters DE, Koh Y, Mitsuya H. Ghosh AK, et al. Among authors: walters de. J Med Chem. 2005 May 19;48(10):3576-85. doi: 10.1021/jm050019i. J Med Chem. 2005. PMID: 15887965

3

Design and synthesis of novel HIV-1 protease inhibitors incorporating oxyindoles as the P2'-ligands.

Ghosh AK, Schiltz G, Perali RS, Leshchenko S, Kay S, Walters DE, Koh Y, Maeda K, Mitsuya H. Ghosh AK, et al. Among authors: walters de. Bioorg Med Chem Lett. 2006 Apr 1;16(7):1869-73. doi: 10.1016/j.bmcl.2006.01.011. Epub 2006 Feb 15. Bioorg Med Chem Lett. 2006. PMID: 16480871

4

Structure-based design of novel HIV-1 protease inhibitors to combat drug resistance.

Ghosh AK, Sridhar PR, Leshchenko S, Hussain AK, Li J, Kovalevsky AY, Walters DE, Wedekind JE, Grum-Tokars V, Das D, Koh Y, Maeda K, Gatanaga H, Weber IT, Mitsuya H. Ghosh AK, et al. Among authors: walters de. J Med Chem. 2006 Aug 24;49(17):5252-61. doi: 10.1021/jm060561m. J Med Chem. 2006. PMID: 16913714

5

Synthesis and biological evaluation of novel allophenylnorstatine-based HIV-1 protease inhibitors incorporating high affinity P2-ligands.

Ghosh AK, Gemma S, Simoni E, Baldridge A, Walters DE, Ide K, Tojo Y, Koh Y, Amano M, Mitsuya H. Ghosh AK, et al. Among authors: walters de. Bioorg Med Chem Lett. 2010 Feb 1;20(3):1241-6. doi: 10.1016/j.bmcl.2009.11.123. Epub 2009 Dec 5. Bioorg Med Chem Lett. 2010. PMID: 20034787 Free PMC article.

6

Potent HIV-1 protease inhibitors incorporating squaramide-derived P2 ligands: Design, synthesis, and biological evaluation.

Ghosh AK, Williams JN, Kovela S, Takayama J, Simpson HM, Walters DE, Hattori SI, Aoki M, Mitsuya H. Ghosh AK, et al. Among authors: walters de. Bioorg Med Chem Lett. 2019 Sep 15;29(18):2565-2570. doi: 10.1016/j.bmcl.2019.08.006. Epub 2019 Aug 5. Bioorg Med Chem Lett. 2019. PMID: 31416666 Free PMC article.

7

Nonpeptidal P2 ligands for HIV protease inhibitors: structure-based design, synthesis, and biological evaluation.

Ghosh AK, Kincaid JF, Walters DE, Chen Y, Chaudhuri NC, Thompson WJ, Culberson C, Fitzgerald PM, Lee HY, McKee SP, Munson PM, Duong TT, Darke PL, Zugay JA, Schleif WA, Axel MG, Lin J, Huff JR. Ghosh AK, et al. Among authors: walters de. J Med Chem. 1996 Aug 16;39(17):3278-90. doi: 10.1021/jm960128k. J Med Chem. 1996. PMID: 8765511

8

Structure based design: novel spirocyclic ethers as nonpeptidal P2-ligands for HIV protease inhibitors.

Ghosh AK, Krishnan K, Walters DE, Cho W, Cho H, Koo Y, Trevino J, Holland L, Buthod J. Ghosh AK, et al. Among authors: walters de. Bioorg Med Chem Lett. 1998 Apr 21;8(8):979-82. doi: 10.1016/s0960-894x(98)00139-5. Bioorg Med Chem Lett. 1998. PMID: 9871524

9

Potent HIV protease inhibitors incorporating high-affinity P2-ligands and (R)-(hydroxyethylamino)sulfonamide isostere.

Ghosh AK, Kincaid JF, Cho W, Walters DE, Krishnan K, Hussain KA, Koo Y, Cho H, Rudall C, Holland L, Buthod J. Ghosh AK, et al. Among authors: walters de. Bioorg Med Chem Lett. 1998 Mar 17;8(6):687-90. doi: 10.1016/s0960-894x(98)00098-5. Bioorg Med Chem Lett. 1998. PMID: 9871583

10

Structure-based design of non-peptide HIV protease inhibitors.

Ghosh AK, Shin D, Swanson L, Krishnan K, Cho H, Hussain KA, Walters DE, Holland L, Buthod J. Ghosh AK, et al. Among authors: walters de. Farmaco. 2001 Jan-Feb;56(1-2):29-32. doi: 10.1016/s0014-827x(01)01025-4. Farmaco. 2001. PMID: 11347961 Review.

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