Espinosa JF - Search Results

1

(2S,1'S,2'S,3'R)-2-(2'-carboxy-3'-methylcyclopropyl) glycine is a potent and selective metabotropic group 2 receptor agonist with anxiolytic properties.

Collado I, Pedregal C, Mazón A, Espinosa JF, Blanco-Urgoiti J, Schoepp DD, Wright RA, Johnson BG, Kingston AE. Collado I, et al. Among authors: espinosa jf. J Med Chem. 2002 Aug 15;45(17):3619-29. doi: 10.1021/jm0110486. J Med Chem. 2002. PMID: 12166935

2

Assignment of absolute configuration on the basis of the conformational effects induced by chiral derivatizing agents: the 2-arylpyrrolidine case.

Vidal P, Pedregal C, Díaz N, Broughton H, Aceña JL, Jiménez A, Espinosa JF. Vidal P, et al. Among authors: espinosa jf. Org Lett. 2007 Oct 11;9(21):4123-6. doi: 10.1021/ol701502e. Epub 2007 Sep 21. Org Lett. 2007. PMID: 17887687

3

Aminoimidazo[1,2-a]pyridines as a new structural class of cyclin-dependent kinase inhibitors. Part 1: Design, synthesis, and biological evaluation.

Jaramillo C, de Diego JE, Hamdouchi C, Collins E, Keyser H, Sánchez-Martínez C, del Prado M, Norman B, Brooks HB, Watkins SA, Spencer CD, Dempsey JA, Anderson BD, Campbell RM, Leggett T, Patel B, Schultz RM, Espinosa J, Vieth M, Zhang F, Timm DE. Jaramillo C, et al. Bioorg Med Chem Lett. 2004 Dec 20;14(24):6095-9. doi: 10.1016/j.bmcl.2004.09.053. Bioorg Med Chem Lett. 2004. PMID: 15546737

4

Preorganization of the hydroxyethylene dipeptide isostere: the preferred conformation in solution resembles the conformation bound to BACE.

Vidal P, Timm D, Broughton H, Chen SH, Martín JA, Rivera-Sagredo A, McCarthy JR, Shapiro MJ, Espinosa JF. Vidal P, et al. Among authors: espinosa jf. J Med Chem. 2005 Dec 1;48(24):7623-7. doi: 10.1021/jm050631+. J Med Chem. 2005. PMID: 16302802

5

Optimization of Hydroxyethylamine Transition State Isosteres as Aspartic Protease Inhibitors by Exploiting Conformational Preferences.

Bueno AB, Agejas J, Broughton H, Dally R, Durham TB, Espinosa JF, González R, Hahn PJ, Marcos A, Rodríguez R, Sanz G, Soriano JF, Timm D, Vidal P, Yang HC, McCarthy JR. Bueno AB, et al. Among authors: espinosa jf. J Med Chem. 2017 Dec 14;60(23):9807-9820. doi: 10.1021/acs.jmedchem.7b01304. Epub 2017 Nov 28. J Med Chem. 2017. PMID: 29088532

6

High resolution magic angle spinning NMR applied to the analysis of organic compounds bound to solid supports.

Espinosa JF. Espinosa JF. Curr Top Med Chem. 2011;11(1):74-92. doi: 10.2174/156802611793611913. Curr Top Med Chem. 2011. PMID: 20809890 Review.

7

Solid-phase synthesis of novel trimers containing a phenylstatine core and analysis by high-resolution magic angle spinning.

Taboada L, Prieto L, Vidal P, Espinosa JF, Erickson JA. Taboada L, et al. Among authors: espinosa jf. J Comb Chem. 2007 Sep-Oct;9(5):748-55. doi: 10.1021/cc070001o. Epub 2007 Jul 14. J Comb Chem. 2007. PMID: 17630807

8

Optimization of diffusion-filtered NMR experiments for selective suppression of residual nondeuterated solvent and water signals from 1H NMR spectra of organic compounds.

Esturau N, Espinosa JF. Esturau N, et al. Among authors: espinosa jf. J Org Chem. 2006 May 26;71(11):4103-10. doi: 10.1021/jo060229i. J Org Chem. 2006. PMID: 16709049

9

A simple method for measuring long-range 1H-13C coupling constants in organic molecules.

Vidal P, Esturau N, Parella T, Espinosa JF. Vidal P, et al. Among authors: espinosa jf. J Org Chem. 2007 Apr 27;72(9):3166-70. doi: 10.1021/jo0621120. Epub 2007 Mar 9. J Org Chem. 2007. PMID: 17346082

10

Conformational features of secondary N-cyclopropyl amides.

González-de-Castro Á, Broughton H, Martínez-Pérez JA, Espinosa JF. González-de-Castro Á, et al. Among authors: espinosa jf. J Org Chem. 2015 Apr 17;80(8):3914-20. doi: 10.1021/acs.joc.5b00236. Epub 2015 Apr 8. J Org Chem. 2015. PMID: 25803271

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