Kafarski P - Search Results

1

Leucine aminopeptidase as a target for inhibitor design.

Grembecka J, Kafarski P. Grembecka J, et al. Among authors: kafarski p. Mini Rev Med Chem. 2001 Jul;1(2):133-44. doi: 10.2174/1389557013406990. Mini Rev Med Chem. 2001. PMID: 12369979 Review.

2

Computer-aided design and activity prediction of leucine aminopeptidase inhibitors.

Grembecka J, Sokalski WA, Kafarski P. Grembecka J, et al. Among authors: kafarski p. J Comput Aided Mol Des. 2000 Aug;14(6):531-44. doi: 10.1023/a:1008189716955. J Comput Aided Mol Des. 2000. PMID: 10921770

3

The most potent organophosphorus inhibitors of leucine aminopeptidase. Structure-based design, chemistry, and activity.

Grembecka J, Mucha A, Cierpicki T, Kafarski P. Grembecka J, et al. Among authors: kafarski p. J Med Chem. 2003 Jun 19;46(13):2641-55. doi: 10.1021/jm030795v. J Med Chem. 2003. PMID: 12801228

4

Stereoselective synthesis of 1-aminoalkanephosphonic acids with two chiral centers and their activity towards leucine aminopeptidase.

Drag M, Pawelczak M, Kafarski P. Drag M, et al. Among authors: kafarski p. Chirality. 2003;15 Suppl:S104-7. doi: 10.1002/chir.10261. Chirality. 2003. PMID: 12884381

5

Synthesis and activity of phosphinic tripeptide inhibitors of cathepsin C.

Mucha A, Paweł M, Hurek J, Kafarski P. Mucha A, et al. Among authors: kafarski p. Bioorg Med Chem Lett. 2004 Jun 21;14(12):3113-6. doi: 10.1016/j.bmcl.2004.04.028. Bioorg Med Chem Lett. 2004. PMID: 15149655

6

alpha-Aminoalkylphosphonates as a tool in experimental optimisation of P1 side chain shape of potential inhibitors in S1 pocket of leucine- and neutral aminopeptidases.

Drag M, Grembecka J, Pawełczak M, Kafarski P. Drag M, et al. Among authors: kafarski p. Eur J Med Chem. 2005 Aug;40(8):764-71. doi: 10.1016/j.ejmech.2005.02.011. Epub 2005 Apr 20. Eur J Med Chem. 2005. PMID: 16122579

7

Design, synthesis, and activity of analogues of phosphinothricin as inhibitors of glutamine synthetase.

Berlicki Ł, Obojska A, Forlani G, Kafarski P. Berlicki Ł, et al. Among authors: kafarski p. J Med Chem. 2005 Oct 6;48(20):6340-9. doi: 10.1021/jm050474e. J Med Chem. 2005. PMID: 16190760

8

Computer-aided analysis of the interactions of glutamine synthetase with its inhibitors.

Berlicki L, Kafarski P. Berlicki L, et al. Among authors: kafarski p. Bioorg Med Chem. 2006 Jul 1;14(13):4578-85. doi: 10.1016/j.bmc.2006.02.022. Epub 2006 Feb 28. Bioorg Med Chem. 2006. PMID: 16504520

9

A phosphonamidate containing aromatic N-terminal amino group as inhibitor of leucine aminopeptidase-design, synthesis and stability.

Mucha A, Kunert A, Grembecka J, Pawełczak M, Kafarski P. Mucha A, et al. Among authors: kafarski p. Eur J Med Chem. 2006 Jun;41(6):768-72. doi: 10.1016/j.ejmech.2006.03.023. Epub 2006 May 11. Eur J Med Chem. 2006. PMID: 16690170

10

Characterization of the Plasmodium falciparum M17 leucyl aminopeptidase. A protease involved in amino acid regulation with potential for antimalarial drug development.

Stack CM, Lowther J, Cunningham E, Donnelly S, Gardiner DL, Trenholme KR, Skinner-Adams TS, Teuscher F, Grembecka J, Mucha A, Kafarski P, Lua L, Bell A, Dalton JP. Stack CM, et al. Among authors: kafarski p. J Biol Chem. 2007 Jan 19;282(3):2069-80. doi: 10.1074/jbc.M609251200. Epub 2006 Nov 15. J Biol Chem. 2007. PMID: 17107951 Free article.

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