Kratzeisen C - Search Results

1

Mutational analysis and molecular modeling of the binding pocket of the metabotropic glutamate 5 receptor negative modulator 2-methyl-6-(phenylethynyl)-pyridine.

Malherbe P, Kratochwil N, Zenner MT, Piussi J, Diener C, Kratzeisen C, Fischer C, Porter RH. Malherbe P, et al. Among authors: kratzeisen c. Mol Pharmacol. 2003 Oct;64(4):823-32. doi: 10.1124/mol.64.4.823. Mol Pharmacol. 2003. PMID: 14500738

2

Mutational analysis and molecular modeling of the allosteric binding site of a novel, selective, noncompetitive antagonist of the metabotropic glutamate 1 receptor.

Malherbe P, Kratochwil N, Knoflach F, Zenner MT, Kew JN, Kratzeisen C, Maerki HP, Adam G, Mutel V. Malherbe P, et al. Among authors: kratzeisen c. J Biol Chem. 2003 Mar 7;278(10):8340-7. doi: 10.1074/jbc.M211759200. Epub 2002 Dec 30. J Biol Chem. 2003. PMID: 12509432 Free article.

3

Identification and characterization of a novel splice variant of the metabotropic glutamate receptor 5 gene in human hippocampus and cerebellum.

Malherbe P, Kew JN, Richards JG, Knoflach F, Kratzeisen C, Zenner MT, Faull RL, Kemp JA, Mutel V. Malherbe P, et al. Among authors: kratzeisen c. Brain Res Mol Brain Res. 2002 Dec 30;109(1-2):168-78. doi: 10.1016/s0169-328x(02)00557-0. Brain Res Mol Brain Res. 2002. PMID: 12531526

4

Opposite effects of Zn on the in vitro binding of [3H]LY354740 to recombinant and native metabotropic glutamate 2 and 3 receptors.

Malherbe P, Richards JG, Broger C, Zenner MT, Messer J, Kratzeisen C, Nakanishi S, Mutel V. Malherbe P, et al. Among authors: kratzeisen c. J Neurochem. 2005 Jul;94(1):150-60. doi: 10.1111/j.1471-4159.2005.03176.x. J Neurochem. 2005. PMID: 15953358 Free article.

5

Me-talnetant and osanetant interact within overlapping but not identical binding pockets in the human tachykinin neurokinin 3 receptor transmembrane domains.

Malherbe P, Bissantz C, Marcuz A, Kratzeisen C, Zenner MT, Wettstein JG, Ratni H, Riemer C, Spooren W. Malherbe P, et al. Among authors: kratzeisen c. Mol Pharmacol. 2008 Jun;73(6):1736-50. doi: 10.1124/mol.107.042754. Epub 2008 Feb 28. Mol Pharmacol. 2008. PMID: 18308898

6

Mapping the binding pocket of dual antagonist almorexant to human orexin 1 and orexin 2 receptors: comparison with the selective OX1 antagonist SB-674042 and the selective OX2 antagonist N-ethyl-2-[(6-methoxy-pyridin-3-yl)-(toluene-2-sulfonyl)-amino]-N-pyridin-3-ylmethyl-acetamide (EMPA).

Malherbe P, Roche O, Marcuz A, Kratzeisen C, Wettstein JG, Bissantz C. Malherbe P, et al. Among authors: kratzeisen c. Mol Pharmacol. 2010 Jul;78(1):81-93. doi: 10.1124/mol.110.064584. Epub 2010 Apr 19. Mol Pharmacol. 2010. PMID: 20404073

7

Identification of essential residues involved in the glutamate binding pocket of the group II metabotropic glutamate receptor.

Malherbe P, Knoflach F, Broger C, Ohresser S, Kratzeisen C, Adam G, Stadler H, Kemp JA, Mutel V. Malherbe P, et al. Among authors: kratzeisen c. Mol Pharmacol. 2001 Nov;60(5):944-54. doi: 10.1124/mol.60.5.944. Mol Pharmacol. 2001. PMID: 11641422

8

Identification of a critical residue in the transmembrane domain 2 of tachykinin neurokinin 3 receptor affecting the dissociation kinetics and antagonism mode of osanetant (SR 142801) and piperidine-based structures.

Malherbe P, Kratzeisen C, Marcuz A, Zenner MT, Nettekoven MH, Ratni H, Wettstein JG, Bissantz C. Malherbe P, et al. Among authors: kratzeisen c. J Med Chem. 2009 Nov 26;52(22):7103-12. doi: 10.1021/jm900948q. J Med Chem. 2009. PMID: 19817444

9

Cloning and functional expression of alternative spliced variants of the human metabotropic glutamate receptor 8.

Malherbe P, Kratzeisen C, Lundstrom K, Richards JG, Faull RL, Mutel V. Malherbe P, et al. Among authors: kratzeisen c. Brain Res Mol Brain Res. 1999 Apr 20;67(2):201-10. doi: 10.1016/s0169-328x(99)00050-9. Brain Res Mol Brain Res. 1999. PMID: 10216218

10

Characterization of (R,S)-5,7-di-tert-butyl-3-hydroxy-3-trifluoromethyl-3H-benzofuran-2-one as a positive allosteric modulator of GABAB receptors.

Malherbe P, Masciadri R, Norcross RD, Knoflach F, Kratzeisen C, Zenner MT, Kolb Y, Marcuz A, Huwyler J, Nakagawa T, Porter RH, Thomas AW, Wettstein JG, Sleight AJ, Spooren W, Prinssen EP. Malherbe P, et al. Among authors: kratzeisen c. Br J Pharmacol. 2008 Jun;154(4):797-811. doi: 10.1038/bjp.2008.135. Epub 2008 Apr 21. Br J Pharmacol. 2008. PMID: 18536733 Free PMC article.

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