Davioud-Charvet E - Search Results

1

Mechanism-based inactivation of thioredoxin reductase from Plasmodium falciparum by Mannich bases. Implication for cytotoxicity.

Davioud-Charvet E, McLeish MJ, Veine DM, Giegel D, Arscott LD, Andricopulo AD, Becker K, Müller S, Schirmer RH, Williams CH Jr, Kenyon GL. Davioud-Charvet E, et al. Biochemistry. 2003 Nov 18;42(45):13319-30. doi: 10.1021/bi0353629. Biochemistry. 2003. PMID: 14609342

2

Specific inhibitors of Plasmodium falciparum thioredoxin reductase as potential antimalarial agents.

Andricopulo AD, Akoachere MB, Krogh R, Nickel C, McLeish MJ, Kenyon GL, Arscott LD, Williams CH Jr, Davioud-Charvet E, Becker K. Andricopulo AD, et al. Bioorg Med Chem Lett. 2006 Apr 15;16(8):2283-92. doi: 10.1016/j.bmcl.2006.01.027. Epub 2006 Feb 3. Bioorg Med Chem Lett. 2006. PMID: 16458512

3

Synthesis of 5,5'-dithiobis(2-nitrobenzamides) as alternative substrates for trypanothione reductase and thioredoxin reductase: a microtiter colorimetric assay for inhibitor screening.

Davioud-Charvet E, Becker K, Landry V, Gromer S, Logé C, Sergheraert C. Davioud-Charvet E, et al. Anal Biochem. 1999 Mar 1;268(1):1-8. doi: 10.1006/abio.1998.3061. Anal Biochem. 1999. PMID: 10036154

4

Mechanistic studies on a novel, highly potent gold-phosphole inhibitor of human glutathione reductase.

Deponte M, Urig S, Arscott LD, Fritz-Wolf K, Réau R, Herold-Mende C, Koncarevic S, Meyer M, Davioud-Charvet E, Ballou DP, Williams CH Jr, Becker K. Deponte M, et al. J Biol Chem. 2005 May 27;280(21):20628-37. doi: 10.1074/jbc.M412519200. Epub 2005 Mar 24. J Biol Chem. 2005. PMID: 15792952 Free article.

5

A prodrug form of a Plasmodium falciparum glutathione reductase inhibitor conjugated with a 4-anilinoquinoline.

Davioud-Charvet E, Delarue S, Biot C, Schwöbel B, Boehme CC, Müssigbrodt A, Maes L, Sergheraert C, Grellier P, Schirmer RH, Becker K. Davioud-Charvet E, et al. J Med Chem. 2001 Nov 22;44(24):4268-76. doi: 10.1021/jm010268g. J Med Chem. 2001. PMID: 11708927

6

5-substituted tetrazoles as bioisosteres of carboxylic acids. Bioisosterism and mechanistic studies on glutathione reductase inhibitors as antimalarials.

Biot C, Bauer H, Schirmer RH, Davioud-Charvet E. Biot C, et al. J Med Chem. 2004 Nov 18;47(24):5972-83. doi: 10.1021/jm0497545. J Med Chem. 2004. PMID: 15537352

7

A fluoro analogue of the menadione derivative 6-[2'-(3'-methyl)-1',4'-naphthoquinolyl]hexanoic acid is a suicide substrate of glutathione reductase. Crystal structure of the alkylated human enzyme.

Bauer H, Fritz-Wolf K, Winzer A, Kühner S, Little S, Yardley V, Vezin H, Palfey B, Schirmer RH, Davioud-Charvet E. Bauer H, et al. J Am Chem Soc. 2006 Aug 23;128(33):10784-94. doi: 10.1021/ja061155v. J Am Chem Soc. 2006. PMID: 16910673

8

Antimalarial dual drugs based on potent inhibitors of glutathione reductase from Plasmodium falciparum.

Friebolin W, Jannack B, Wenzel N, Furrer J, Oeser T, Sanchez CP, Lanzer M, Yardley V, Becker K, Davioud-Charvet E. Friebolin W, et al. J Med Chem. 2008 Mar 13;51(5):1260-77. doi: 10.1021/jm7009292. Epub 2008 Feb 9. J Med Chem. 2008. PMID: 18260613

9

Glutathione reductase-catalyzed cascade of redox reactions to bioactivate potent antimalarial 1,4-naphthoquinones--a new strategy to combat malarial parasites.

Müller T, Johann L, Jannack B, Brückner M, Lanfranchi DA, Bauer H, Sanchez C, Yardley V, Deregnaucourt C, Schrével J, Lanzer M, Schirmer RH, Davioud-Charvet E. Müller T, et al. J Am Chem Soc. 2011 Aug 3;133(30):11557-71. doi: 10.1021/ja201729z. Epub 2011 Jul 12. J Am Chem Soc. 2011. PMID: 21682307

10

Synthesis of 5-nitro-2-furancarbohydrazides and their cis-diamminedichloroplatinum complexes as bitopic and irreversible human thioredoxin reductase inhibitors.

Millet R, Urig S, Jacob J, Amtmann E, Moulinoux JP, Gromer S, Becker K, Davioud-Charvet E. Millet R, et al. J Med Chem. 2005 Nov 3;48(22):7024-39. doi: 10.1021/jm050256l. J Med Chem. 2005. PMID: 16250662

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