Guillon G - Search Results

1

The discovery of novel vasopressin V1b receptor ligands for pharmacological, functional and structural investigations.

Guillon G, Derick S, Pena A, Cheng LL, Stoev S, Seyer R, Morgat JL, Barberis C, Gal CS, Wagnon J, Manning M. Guillon G, et al. J Neuroendocrinol. 2004 Apr;16(4):356-61. doi: 10.1111/j.0953-8194.2004.01163.x. J Neuroendocrinol. 2004. PMID: 15089974 Review.

2

[1-deamino-4-cyclohexylalanine] arginine vasopressin: a potent and specific agonist for vasopressin V1b receptors.

Derick S, Cheng LL, Voirol MJ, Stoev S, Giacomini M, Wo NC, Szeto HH, Ben Mimoun M, Andres M, Gaillard RC, Guillon G, Manning M. Derick S, et al. Among authors: guillon g. Endocrinology. 2002 Dec;143(12):4655-64. doi: 10.1210/en.2002-220363. Endocrinology. 2002. PMID: 12446593

3

Key amino acids located within the transmembrane domains 5 and 7 account for the pharmacological specificity of the human V1b vasopressin receptor.

Derick S, Pena A, Durroux T, Wagnon J, Serradeil-Le Gal C, Hibert M, Rognan D, Guillon G. Derick S, et al. Among authors: guillon g. Mol Endocrinol. 2004 Nov;18(11):2777-89. doi: 10.1210/me.2004-0124. Epub 2004 Jul 29. Mol Endocrinol. 2004. PMID: 15284336

4

Characterization of (2S,4R)-1-[5-chloro-1-[(2,4-dimethoxyphenyl)sulfonyl]-3-(2-methoxy-phenyl)-2-oxo-2,3-dihydro-1H-indol-3-yl]-4-hydroxy-N,N-dimethyl-2-pyrrolidine carboxamide (SSR149415), a selective and orally active vasopressin V1b receptor antagonist.

Serradeil-Le Gal C, Wagnon J, Simiand J, Griebel G, Lacour C, Guillon G, Barberis C, Brossard G, Soubrié P, Nisato D, Pascal M, Pruss R, Scatton B, Maffrand JP, Le Fur G. Serradeil-Le Gal C, et al. Among authors: guillon g. J Pharmacol Exp Ther. 2002 Mar;300(3):1122-30. doi: 10.1124/jpet.300.3.1122. J Pharmacol Exp Ther. 2002. PMID: 11861823

5

Functional and pharmacological characterization of the first specific agonist and antagonist for the V1b receptor in mammals.

Serradeil-Le Gal C, Derick S, Brossard G, Manning M, Simiand J, Gaillard R, Griebel G, Guillon G. Serradeil-Le Gal C, et al. Among authors: guillon g. Stress. 2003 Sep;6(3):199-206. doi: 10.1080/1025389032000114524. Stress. 2003. PMID: 13129813 Free article. Review.

6

Design of potent and selective agonists for the human vasopressin V1b receptor based on modifications of [deamino-cys1]arginine vasopressin at position 4.

Cheng LL, Stoev S, Manning M, Derick S, Pena A, Mimoun MB, Guillon G. Cheng LL, et al. Among authors: guillon g. J Med Chem. 2004 Apr 22;47(9):2375-88. doi: 10.1021/jm030611c. J Med Chem. 2004. PMID: 15084136

7

Comparative pharmacology of bovine, human and rat vasopressin receptor isoforms.

Andrés M, Peña A, Derick S, Raufaste D, Trojnar J, Wisniewski K, Trueba M, Serradeil-Le Gal C, Guillon G. Andrés M, et al. Among authors: guillon g. Eur J Pharmacol. 2004 Oct 6;501(1-3):59-69. doi: 10.1016/j.ejphar.2004.08.026. Eur J Pharmacol. 2004. PMID: 15464063

8

Position 4 analogues of [deamino-Cys(1)] arginine vasopressin exhibit striking species differences for human and rat V(2)/V(1b) receptor selectivity.

Guillon G, Pena A, Murat B, Derick S, Trueba M, Ventura MA, Szeto HH, Wo N, Stoev S, Cheng LL, Manning M. Guillon G, et al. J Pept Sci. 2006 Mar;12(3):190-8. doi: 10.1002/psc.710. J Pept Sci. 2006. PMID: 16130178

9

Design and synthesis of the first selective agonists for the rat vasopressin V(1b) receptor: based on modifications of deamino-[Cys1]arginine vasopressin at positions 4 and 8.

Pena A, Murat B, Trueba M, Ventura MA, Wo NC, Szeto HH, Cheng LL, Stoev S, Guillon G, Manning M. Pena A, et al. Among authors: guillon g. J Med Chem. 2007 Feb 22;50(4):835-47. doi: 10.1021/jm060928n. J Med Chem. 2007. PMID: 17300166

10

Pharmacological and physiological characterization of d[Leu4, Lys8]vasopressin, the first V1b-selective agonist for rat vasopressin/oxytocin receptors.

Pena A, Murat B, Trueba M, Ventura MA, Bertrand G, Cheng LL, Stoev S, Szeto HH, Wo N, Brossard G, Serradeil-Le Gal C, Manning M, Guillon G. Pena A, et al. Among authors: guillon g. Endocrinology. 2007 Sep;148(9):4136-46. doi: 10.1210/en.2006-1633. Epub 2007 May 10. Endocrinology. 2007. PMID: 17495006

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