Perregaard J - Search Results

1

First demonstration of a functional role for central nervous system betaine/{gamma}-aminobutyric acid transporter (mGAT2) based on synergistic anticonvulsant action among inhibitors of mGAT1 and mGAT2.

White HS, Watson WP, Hansen SL, Slough S, Perregaard J, Sarup A, Bolvig T, Petersen G, Larsson OM, Clausen RP, Frølund B, Falch E, Krogsgaard-Larsen P, Schousboe A. White HS, et al. Among authors: perregaard j. J Pharmacol Exp Ther. 2005 Feb;312(2):866-74. doi: 10.1124/jpet.104.068825. Epub 2004 Nov 18. J Pharmacol Exp Ther. 2005. PMID: 15550575

2

Selective inhibitors of GABA uptake: synthesis and molecular pharmacology of 4-N-methylamino-4,5,6,7-tetrahydrobenzo[d]isoxazol-3-ol analogues.

Clausen RP, Moltzen EK, Perregaard J, Lenz SM, Sanchez C, Falch E, Frølund B, Bolvig T, Sarup A, Larsson OM, Schousboe A, Krogsgaard-Larsen P. Clausen RP, et al. Among authors: perregaard j. Bioorg Med Chem. 2005 Feb 1;13(3):895-908. doi: 10.1016/j.bmc.2004.10.029. Bioorg Med Chem. 2005. PMID: 15653355

3

Selective inhibitors of glial GABA uptake: synthesis, absolute stereochemistry, and pharmacology of the enantiomers of 3-hydroxy-4-amino-4,5,6,7-tetrahydro-1,2-benzisoxazole (exo-THPO) and analogues.

Falch E, Perregaard J, FrŁlund B, SŁkilde B, Buur A, Hansen LM, Frydenvang K, Brehm L, Bolvig T, Larsson OM, Sanchez C, White HS, Schousboe A, Krogsgaard-Larsen P. Falch E, et al. Among authors: perregaard j. J Med Chem. 1999 Dec 30;42(26):5402-14. doi: 10.1021/jm9904452. J Med Chem. 1999. PMID: 10639282

4

The selective sigma2-ligand Lu 28-179 has potent anxiolytic-like effects in rodents.

Sánchez C, Arnt J, Costall B, Kelly ME, Meier E, Naylor RJ, Perregaard J. Sánchez C, et al. Among authors: perregaard j. J Pharmacol Exp Ther. 1997 Dec;283(3):1323-32. J Pharmacol Exp Ther. 1997. PMID: 9400007

5

Selective, centrally acting serotonin 5-HT2 antagonists. 1. 2- and 6-substituted 1-phenyl-3-(4-piperidinyl)-1H-indoles.

Perregaard J, Andersen K, Hyttel J, Sánchez C. Perregaard J, et al. J Med Chem. 1992 Dec 25;35(26):4813-22. doi: 10.1021/jm00104a006. J Med Chem. 1992. PMID: 1336053

6

Noncataleptogenic, centrally acting dopamine D-2 and serotonin 5-HT2 antagonists within a series of 3-substituted 1-(4-fluorophenyl)-1H-indoles.

Perregaard J, Arnt J, Bøgesø KP, Hyttel J, Sánchez C. Perregaard J, et al. J Med Chem. 1992 Mar 20;35(6):1092-101. doi: 10.1021/jm00084a014. J Med Chem. 1992. PMID: 1348090

7

Sigma ligands with subnanomolar affinity and preference for the sigma 2 binding site. 1. 3-(omega-aminoalkyl)-1H-indoles.

Perregaard J, Moltzen EK, Meier E, Sánchez C. Perregaard J, et al. J Med Chem. 1995 May 26;38(11):1998-2008. doi: 10.1021/jm00011a019. J Med Chem. 1995. PMID: 7783131

8

Sigma ligands with subnanomolar affinity and preference for the sigma 2 binding site. 2. Spiro-joined benzofuran, isobenzofuran, and benzopyran piperidines.

Moltzen EK, Perregaard J, Meier E. Moltzen EK, et al. Among authors: perregaard j. J Med Chem. 1995 May 26;38(11):2009-17. doi: 10.1021/jm00011a020. J Med Chem. 1995. PMID: 7783132

9

Synthesis and structure-affinity relationship investigations of 5-aminomethyl and 5-carbamoyl analogues of the antipsychotic sertindole. A new class of selective alpha1 adrenoceptor antagonists.

Balle T, Perregaard J, Larsen AK, Ramirez MT, Krøjer Søby K, Liljefors T, Andersen K. Balle T, et al. Among authors: perregaard j. Bioorg Med Chem. 2003 Mar 20;11(6):1065-78. doi: 10.1016/s0968-0896(02)00459-5. Bioorg Med Chem. 2003. PMID: 12614894

10

Synthesis and structure-affinity relationship investigations of 5-heteroaryl-substituted analogues of the antipsychotic sertindole. A new class of highly selective alpha(1) adrenoceptor antagonists.

Balle T, Perregaard J, Ramirez MT, Larsen AK, Søby KK, Liljefors T, Andersen K. Balle T, et al. Among authors: perregaard j. J Med Chem. 2003 Jan 16;46(2):265-83. doi: 10.1021/jm020938y. J Med Chem. 2003. PMID: 12519065

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