Trapani G - Search Results

1

Structure-activity relationships and effects on neuroactive steroid synthesis in a series of 2-phenylimidazo[1,2-a]pyridineacetamide peripheral benzodiazepine receptors ligands.

Trapani G, Laquintana V, Denora N, Trapani A, Lopedota A, Latrofa A, Franco M, Serra M, Pisu MG, Floris I, Sanna E, Biggio G, Liso G. Trapani G, et al. Among authors: trapani a. J Med Chem. 2005 Jan 13;48(1):292-305. doi: 10.1021/jm049610q. J Med Chem. 2005. PMID: 15634024

2

Synthesis and pharmacological evaluation of 1-[(1,2-diphenyl-1H-4-imidazolyl)methyl]-4-phenylpiperazines with clozapine-like mixed activities at dopamine D(2), serotonin, and GABA(A) receptors.

Asproni B, Pau A, Bitti M, Melosu M, Cerri R, Dazzi L, Seu E, Maciocco E, Sanna E, Busonero F, Talani G, Pusceddu L, Altomare C, Trapani G, Biggio G. Asproni B, et al. Among authors: trapani g. J Med Chem. 2002 Oct 10;45(21):4655-68. doi: 10.1021/jm020848t. J Med Chem. 2002. PMID: 12361392

3

Peripheral benzodiazepine receptor ligand-melphalan conjugates for potential selective drug delivery to brain tumors.

Trapani G, Laquintana V, Latrofa A, Ma J, Reed K, Serra M, Biggio G, Liso G, Gallo JM. Trapani G, et al. Bioconjug Chem. 2003 Jul-Aug;14(4):830-9. doi: 10.1021/bc034023p. Bioconjug Chem. 2003. PMID: 12862438

4

Synthesis and characterization of a platinum(II) complex tethered to a ligand of the peripheral benzodiazepine receptor.

Margiotta N, Ostuni R, Ranaldo R, Denora N, Laquintana V, Trapani G, Liso G, Natile G. Margiotta N, et al. Among authors: trapani g. J Med Chem. 2007 Mar 8;50(5):1019-27. doi: 10.1021/jm0612160. Epub 2007 Feb 8. J Med Chem. 2007. PMID: 17286392

5

N-benzyl-2-(6,8-dichloro-2-(4-chlorophenyl)imidazo[1,2-a]pyridin-3-yl)-N-(6-(7-nitrobenzo[c][1,2,5]oxadiazol-4-ylamino)hexyl)acetamide as a new fluorescent probe for peripheral benzodiazepine receptor and microglial cell visualization.

Laquintana V, Denora N, Lopedota A, Suzuki H, Sawada M, Serra M, Biggio G, Latrofa A, Trapani G, Liso G. Laquintana V, et al. Among authors: trapani g. Bioconjug Chem. 2007 Sep-Oct;18(5):1397-407. doi: 10.1021/bc060393c. Epub 2007 Aug 28. Bioconjug Chem. 2007. PMID: 17722875

6

2-Phenyl-imidazo[1,2-a]pyridine compounds containing hydrophilic groups as potent and selective ligands for peripheral benzodiazepine receptors: synthesis, binding affinity and electrophysiological studies.

Denora N, Laquintana V, Pisu MG, Dore R, Murru L, Latrofa A, Trapani G, Sanna E. Denora N, et al. Among authors: trapani g. J Med Chem. 2008 Nov 13;51(21):6876-88. doi: 10.1021/jm8006728. Epub 2008 Oct 4. J Med Chem. 2008. PMID: 18834105

7

Recent advances in medicinal chemistry and pharmaceutical technology--strategies for drug delivery to the brain.

Denora N, Trapani A, Laquintana V, Lopedota A, Trapani G. Denora N, et al. Among authors: trapani g, trapani a. Curr Top Med Chem. 2009;9(2):182-96. doi: 10.2174/156802609787521571. Curr Top Med Chem. 2009. PMID: 19200004 Review.

8

Platinum(II) complexes with bioactive carrier ligands having high affinity for the translocator protein.

Margiotta N, Denora N, Ostuni R, Laquintana V, Anderson A, Johnson SW, Trapani G, Natile G. Margiotta N, et al. Among authors: trapani g. J Med Chem. 2010 Jul 22;53(14):5144-54. doi: 10.1021/jm100429r. J Med Chem. 2010. PMID: 20568783

9

Synthesis and binding affinity of 2-phenylimidazo[1,2-alpha]pyridine derivatives for both central and peripheral benzodiazepine receptors. A new series of high-affinity and selective ligands for the peripheral type.

Trapani G, Franco M, Ricciardi L, Latrofa A, Genchi G, Sanna E, Tuveri F, Cagetti E, Biggio G, Liso G. Trapani G, et al. J Med Chem. 1997 Sep 12;40(19):3109-18. doi: 10.1021/jm970112+. J Med Chem. 1997. PMID: 9301675

10

Propofol analogues. Synthesis, relationships between structure and affinity at GABAA receptor in rat brain, and differential electrophysiological profile at recombinant human GABAA receptors.

Trapani G, Latrofa A, Franco M, Altomare C, Sanna E, Usala M, Biggio G, Liso G. Trapani G, et al. J Med Chem. 1998 May 21;41(11):1846-54. doi: 10.1021/jm970681h. J Med Chem. 1998. PMID: 9599235

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