Neamati N - Search Results

1

Design of novel bioisosteres of beta-diketo acid inhibitors of HIV-1 integrase.

Sechi M, Sannia L, Carta F, Palomba M, Dallocchio R, Dessì A, Derudas M, Zawahir Z, Neamati N. Sechi M, et al. Among authors: neamati n. Antivir Chem Chemother. 2005;16(1):41-61. doi: 10.1177/095632020501600105. Antivir Chem Chemother. 2005. PMID: 15739621 Free article.

2

Design and synthesis of novel dihydroxyindole-2-carboxylic acids as HIV-1 integrase inhibitors.

Sechi M, Angotzi G, Dallocchio R, Dessì A, Carta F, Sannia L, Mariani A, Fiori S, Sanchez T, Movsessian L, Plasencia C, Neamati N. Sechi M, et al. Among authors: neamati n. Antivir Chem Chemother. 2004 Mar;15(2):67-81. doi: 10.1177/095632020401500203. Antivir Chem Chemother. 2004. PMID: 15185725 Free article.

3

Design and synthesis of novel indole beta-diketo acid derivatives as HIV-1 integrase inhibitors.

Sechi M, Derudas M, Dallocchio R, Dessì A, Bacchi A, Sannia L, Carta F, Palomba M, Ragab O, Chan C, Shoemaker R, Sei S, Dayam R, Neamati N. Sechi M, et al. Among authors: neamati n. J Med Chem. 2004 Oct 7;47(21):5298-310. doi: 10.1021/jm049944f. J Med Chem. 2004. PMID: 15456274

A plethora of diketo acid-containing compounds have been claimed in patent literature without disclosing much biological activities and synthetic details (reviewed in Neamati, N. Exp. Opin. Ther. Pat. 2002, 12, 709-724). To establish a coherent structure-activity re …

A plethora of diketo acid-containing compounds have been claimed in patent literature without disclosing much biological activities and synt …

4

From ligand to complexes: inhibition of human immunodeficiency virus type 1 integrase by beta-diketo acid metal complexes.

Sechi M, Bacchi A, Carcelli M, Compari C, Duce E, Fisicaro E, Rogolino D, Gates P, Derudas M, Al-Mawsawi LQ, Neamati N. Sechi M, et al. Among authors: neamati n. J Med Chem. 2006 Jul 13;49(14):4248-60. doi: 10.1021/jm060193m. J Med Chem. 2006. PMID: 16821784

5

Design and synthesis of bis-amide and hydrazide-containing derivatives of malonic acid as potential HIV-1 integrase inhibitors.

Sechi M, Azzena U, Delussu MP, Dallocchio R, Dessì A, Cosseddu A, Pala N, Neamati N. Sechi M, et al. Among authors: neamati n. Molecules. 2008 Oct 1;13(10):2442-61. doi: 10.3390/molecules13102442. Molecules. 2008. PMID: 18830166 Free PMC article.

6

From ligand to complexes. Part 2. Remarks on human immunodeficiency virus type 1 integrase inhibition by beta-diketo acid metal complexes.

Bacchi A, Biemmi M, Carcelli M, Carta F, Compari C, Fisicaro E, Rogolino D, Sechi M, Sippel M, Sotriffer CA, Sanchez TW, Neamati N. Bacchi A, et al. Among authors: neamati n. J Med Chem. 2008 Nov 27;51(22):7253-64. doi: 10.1021/jm800893q. J Med Chem. 2008. PMID: 18983138

7

Design and synthesis of novel dihydroquinoline-3-carboxylic acids as HIV-1 integrase inhibitors.

Sechi M, Rizzi G, Bacchi A, Carcelli M, Rogolino D, Pala N, Sanchez TW, Taheri L, Dayam R, Neamati N. Sechi M, et al. Among authors: neamati n. Bioorg Med Chem. 2009 Apr 1;17(7):2925-35. doi: 10.1016/j.bmc.2008.10.088. Epub 2008 Nov 6. Bioorg Med Chem. 2009. PMID: 19026554

8

Design, synthesis, molecular modeling, and anti-HIV-1 integrase activity of a series of photoactivatable diketo acid-containing inhibitors as affinity probes.

Sechi M, Carta F, Sannia L, Dallocchio R, Dessì A, Al-Safi RI, Neamati N. Sechi M, et al. Among authors: neamati n. Antiviral Res. 2009 Mar;81(3):267-76. doi: 10.1016/j.antiviral.2008.12.010. Epub 2009 Jan 9. Antiviral Res. 2009. PMID: 19135482

9

Sequence-based design and discovery of peptide inhibitors of HIV-1 integrase: insight into the binding mode of the enzyme.

Li HY, Zawahir Z, Song LD, Long YQ, Neamati N. Li HY, et al. Among authors: neamati n. J Med Chem. 2006 Jul 27;49(15):4477-86. doi: 10.1021/jm060307u. J Med Chem. 2006. PMID: 16854053

10

Inhibition of HIV-1 integrase activity by synthetic peptides derived from the HIV-1 HXB2 Pol region of the viral genome.

Zawahir Z, Neamati N. Zawahir Z, et al. Among authors: neamati n. Bioorg Med Chem Lett. 2006 Oct 1;16(19):5199-202. doi: 10.1016/j.bmcl.2006.07.022. Epub 2006 Aug 1. Bioorg Med Chem Lett. 2006. PMID: 16879966

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