Lescot E - Search Results

1

3D-QSAR and docking studies of selective GSK-3beta inhibitors. Comparison with a thieno[2,3-b]pyrrolizinone derivative, a new potential lead for GSK-3beta ligands.

Lescot E, Bureau R, Sopkova-de Oliveira Santos J, Rochais C, Lisowski V, Lancelot JC, Rault S. Lescot E, et al. J Chem Inf Model. 2005 May-Jun;45(3):708-15. doi: 10.1021/ci050008y. J Chem Inf Model. 2005. PMID: 15921460

2

Synthesis and biological evaluation of thienopyrrolizines, a new family of CDK/GSK-3 inhibitors.

Rochais C, Lescot E, Lisowski V, Lepailleur A, Santos JS, Bureau R, Dallemagne P, Meijer L, Rault S. Rochais C, et al. Among authors: lescot e. J Enzyme Inhib Med Chem. 2004 Dec;19(6):585-93. doi: 10.1080/14756360400004565. J Enzyme Inhib Med Chem. 2004. PMID: 15662962 Free article.

3

Definition of new pharmacophores for nonpeptide antagonists of human urotensin-II. Comparison with the 3D-structure of human urotensin-II and URP.

Lescot E, Sopkova-de Oliveira Santos J, Dubessy C, Oulyadi H, Lesnard A, Vaudry H, Bureau R, Rault S. Lescot E, et al. J Chem Inf Model. 2007 Mar-Apr;47(2):602-12. doi: 10.1021/ci6003948. J Chem Inf Model. 2007. PMID: 17381176

4

Synthesis of new dipyrrolo- and furopyrrolopyrazinones related to tripentones and their biological evaluation as potential kinases (CDKs1-5, GSK-3) inhibitors.

Rochais C, Duc NV, Lescot E, Sopkova-de Oliveira Santos J, Bureau R, Meijer L, Dallemagne P, Rault S. Rochais C, et al. Among authors: lescot e. Eur J Med Chem. 2009 Feb;44(2):708-16. doi: 10.1016/j.ejmech.2008.05.011. Epub 2008 May 23. Eur J Med Chem. 2009. PMID: 18586356

5

Synthesis and biological evaluation as AChE inhibitors of new indanones and thiaindanones related to donepezil.

Omran Z, Cailly T, Lescot E, Santos JS, Agondanou JH, Lisowski V, Fabis F, Godard AM, Stiebing S, Le Flem G, Boulouard M, Dauphin F, Dallemagne P, Rault S. Omran Z, et al. Among authors: lescot e. Eur J Med Chem. 2005 Dec;40(12):1222-45. doi: 10.1016/j.ejmech.2005.07.009. Epub 2005 Aug 30. Eur J Med Chem. 2005. PMID: 16137794

6

Nonpeptide Urotensin-II receptor agonists and antagonists: review and structure-activity relationships.

Lescot E, Bureau R, Rault S. Lescot E, et al. Peptides. 2008 May;29(5):680-90. doi: 10.1016/j.peptides.2007.09.019. Epub 2007 Oct 6. Peptides. 2008. PMID: 18022732 Review.

7

Three-dimensional model of the human urotensin-II receptor: docking of human urotensin-II and nonpeptide antagonists in the binding site and comparison with an antagonist pharmacophore model.

Lescot E, Sopkova-de Oliveira Santos J, Colloc'h N, Rodrigo J, Milazzo-Segalas I, Bureau R, Rault S. Lescot E, et al. Proteins. 2008 Oct;73(1):173-84. doi: 10.1002/prot.22050. Proteins. 2008. PMID: 18409194

8

Prediction of acute toxicity in fish by using QSAR methods and chemical modes of action.

Lozano S, Lescot E, Halm MP, Lepailleur A, Bureau R, Rault S. Lozano S, et al. Among authors: lescot e. J Enzyme Inhib Med Chem. 2010 Apr;25(2):195-203. doi: 10.3109/14756360903169857. J Enzyme Inhib Med Chem. 2010. PMID: 19874208 Free article.

9

DNA-drug recognition and effects on topoisomerase II-mediated cytotoxicity. A three-mode binding model for ellipticine derivatives.

Monnot M, Mauffret O, Simon V, Lescot E, Psaume B, Saucier JM, Charra M, Belehradek J Jr, Fermandjian S. Monnot M, et al. Among authors: lescot e. J Biol Chem. 1991 Jan 25;266(3):1820-9. J Biol Chem. 1991. PMID: 1846365 Free article.

10

Synthesis of 11H-pyridocarbazoles and derivatives. Comparison of their DNA binding and antitumor activity with those of 6H- and 7H-pyridocarbazoles.

Lescot E, Muzard G, Markovits J, Belleney J, Roques BP, Le Pecq JB. Lescot E, et al. J Med Chem. 1986 Sep;29(9):1731-7. doi: 10.1021/jm00159a028. J Med Chem. 1986. PMID: 3746819

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