Vaz RJ - Search Results

1

Discovery of novel 1-arylmethyl pyrrolidin-2-yl ethanol amines as calcium-sensing receptor antagonists.

Gavai AV, Vaz RJ, Mikkilineni AB, Roberge JY, Liu Y, Lawrence RM, Corte JR, Yang W, Bednarz M, Dickson JK Jr, Ma Z, Seethala R, Feyen JH. Gavai AV, et al. Among authors: vaz rj. Bioorg Med Chem Lett. 2005 Dec 15;15(24):5478-82. doi: 10.1016/j.bmcl.2005.08.095. Epub 2005 Oct 10. Bioorg Med Chem Lett. 2005. PMID: 16216508

2

A 3D-QSAR model for CYP2D6 inhibition in the aryloxypropanolamine series.

Vaz RJ, Nayeem A, Santone K, Chandrasena G, Gavai AV. Vaz RJ, et al. Bioorg Med Chem Lett. 2005 Sep 1;15(17):3816-20. doi: 10.1016/j.bmcl.2005.06.007. Bioorg Med Chem Lett. 2005. PMID: 15993593

3

Design and synthesis of a G-protein-coupled receptor antagonist library of aryloxyalkanolamines using a polymer-supported acyclic acetal linker.

Roberge JY, Harikrishnan LS, Kamau MG, Ruan Z, Van Kirk K, Liu Y, Cooper CB, Poss MA, Dickson JK Jr, Gavai AV, Chao ST, Leith LW, Bednarz MS, Mathur A, Kakarla R, Schnur DM, Vaz R, Lawrence RM. Roberge JY, et al. J Comb Chem. 2009 Jan-Feb;11(1):72-82. doi: 10.1021/cc800051u. J Comb Chem. 2009. PMID: 19086798

4

Characterization of HERG potassium channel inhibition using CoMSiA 3D QSAR and homology modeling approaches.

Pearlstein RA, Vaz RJ, Kang J, Chen XL, Preobrazhenskaya M, Shchekotikhin AE, Korolev AM, Lysenkova LN, Miroshnikova OV, Hendrix J, Rampe D. Pearlstein RA, et al. Among authors: vaz rj. Bioorg Med Chem Lett. 2003 May 19;13(10):1829-35. doi: 10.1016/s0960-894x(03)00196-3. Bioorg Med Chem Lett. 2003. PMID: 12729675

5

Design, synthesis, and biological activity of potent and selective inhibitors of mast cell tryptase.

Hopkins CR, Czekaj M, Kaye SS, Gao Z, Pribish J, Pauls H, Liang G, Sides K, Cramer D, Cairns J, Luo Y, Lim HK, Vaz R, Rebello S, Maignan S, Dupuy A, Mathieu M, Levell J. Hopkins CR, et al. Bioorg Med Chem Lett. 2005 Jun 2;15(11):2734-7. doi: 10.1016/j.bmcl.2005.04.002. Bioorg Med Chem Lett. 2005. PMID: 15911249

6

Design of bivalent ligands using hydrogen bond linkers: synthesis and evaluation of inhibitors for human beta-tryptase.

Vaz RJ, Gao Z, Pribish J, Chen X, Levell J, Davis L, Albert E, Brollo M, Ugolini A, Cramer DM, Cairns J, Sides K, Liu F, Kwong J, Kang J, Rebello S, Elliot M, Lim H, Chellaraj V, Singleton RW, Li Y. Vaz RJ, et al. Bioorg Med Chem Lett. 2004 Dec 20;14(24):6053-6. doi: 10.1016/j.bmcl.2004.09.065. Bioorg Med Chem Lett. 2004. PMID: 15546728

7

Discovery of covalent inhibitors for MIF tautomerase via cocrystal structures with phantom hits from virtual screening.

McLean LR, Zhang Y, Li H, Li Z, Lukasczyk U, Choi YM, Han Z, Prisco J, Fordham J, Tsay JT, Reiling S, Vaz RJ, Li Y. McLean LR, et al. Among authors: vaz rj. Bioorg Med Chem Lett. 2009 Dec 1;19(23):6717-20. doi: 10.1016/j.bmcl.2009.09.106. Epub 2009 Oct 1. Bioorg Med Chem Lett. 2009. PMID: 19836948

8

Discovery of novel inhibitors for DHODH via virtual screening and X-ray crystallographic structures.

McLean LR, Zhang Y, Degnen W, Peppard J, Cabel D, Zou C, Tsay JT, Subramaniam A, Vaz RJ, Li Y. McLean LR, et al. Among authors: vaz rj. Bioorg Med Chem Lett. 2010 Mar 15;20(6):1981-4. doi: 10.1016/j.bmcl.2010.01.115. Epub 2010 Jan 25. Bioorg Med Chem Lett. 2010. PMID: 20153645

9

Novel steroidal vinyl fluorides as inhibitors of steroid C17(20) lyase.

Burkhart JP, Weintraub PM, Gates CA, Resvick RJ, Vaz RJ, Friedrich D, Angelastro MR, Bey P, Peet NP. Burkhart JP, et al. Among authors: vaz rj. Bioorg Med Chem. 2002 Apr;10(4):929-34. doi: 10.1016/s0968-0896(01)00354-6. Bioorg Med Chem. 2002. PMID: 11836100

10

Understanding DP receptor antagonism using a CoMSIA approach.

Mu L, Aguiar J, Ardati A, Cao B, Gardner CJ, Gillespy T, Harris K, Lim S, Marcus R, Morize I, Parkar A, Stefany D, Li Y, Vaz RJ, Cirovic DA. Mu L, et al. Among authors: vaz rj. Bioorg Med Chem Lett. 2011 Jan 1;21(1):66-75. doi: 10.1016/j.bmcl.2010.11.071. Epub 2010 Nov 21. Bioorg Med Chem Lett. 2011. PMID: 21147533

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